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7-(3-hydroxypyridine-2-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-3-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]urea
3-cyclohexyl-4-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
5-chloro-3-fluoro-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]pyridine
2-{1-[(2,3,4-trimethoxyphenyl)methyl]pyrrolidin-2-yl}-1,3-thiazole
4-[(1R,7S)-3-tert-butyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carbonyl]-1λ6-thiomorpholine-1,1-dione
N-(4-chloro-2-fluorophenyl)-2-{methyl[3-(oxolan-2-yl)propyl]amino}acetamide
2-(3-{[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}phenoxymethyl)pyridine
1-[2-(3-fluorophenyl)piperidin-1-yl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
2-(2-fluorophenyl)-2-{[4-(piperidin-1-ylmethyl)phenyl]formamido}acetic acid
7-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-4-(2-oxopyrrolidin-1-yl)benzamide
4-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
4-[4-ethyl-6-(pyridin-3-yl)pyrimidin-2-yl]morpholine
2-(dimethylamino)-4-methyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrimidine-5-carboxamide
6-methyl-2-(pyridin-3-yl)-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]pyrimidin-4-amine
1-[(2R)-pyrrolidine-2-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(2,3-dimethylphenyl)-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]acetic acid
methyl 6-[2-(3-fluorophenyl)acetyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-cycloheptyl-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-[1-methyl-4-(3,3,3-trifluoropropyl)-1,4,9-triazaspiro[5.5]undecan-9-yl]-2-phenoxyethan-1-one
5-ethyl-2-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
7-[(2,3-difluorophenyl)methyl]-N-ethyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-3-acetamido-N-methylthiophene-2-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-(furan-2-carbonyl)-3-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}piperidine
1-(3-methoxyphenyl)-4-[(2S)-2-(methylamino)propanoyl]piperazin-2-one
N-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(4-chlorophenyl)methyl]-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
methyl 2-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}-1,3-oxazole-4-carboxylate
7-(2-methylphenyl)-4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[2-(pyrrolidin-1-yl)ethyl]-1-{4-[(trifluoromethyl)sulfanyl]phenyl}urea
3-[({[2-(2-methylpropoxy)phenyl]carbamoyl}amino)methyl]-1,2,4-oxadiazole-5-carboxamide
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-1-(4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
N-[1-(2-methylpropanoyl)piperidin-3-yl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
[(3R,4R)-1-(3-chloro-4-fluorobenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
6-methyl-2-({2-oxo-2-[3-(1H-pyrazol-3-yl)piperidin-1-yl]ethyl}sulfanyl)-3,4-dihydropyrimidin-4-one
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
8-(3-hydroxy-4-methylbenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(2,2-difluoroethyl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
(1R,5R)-6-(cyclopropylmethyl)-N-(2-ethoxyphenyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(1S,5R)-6-(1H-imidazol-2-ylmethyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(3R,9aR)-3-benzyl-8-[(3-chlorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[(3R,4S)-1-(2-amino-6-methoxypyrimidin-4-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1-[(3S)-1-benzylpiperidin-3-yl]-3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}urea
N3-methyl-N3-(quinoxalin-2-ylmethyl)piperidine-1,3-dicarboxamide
1-[5-(2-methylbenzenesulfonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]pyrrolidine
N-[(4-chlorophenyl)methyl]-3-(hydroxymethyl)-3-(3-methoxypropyl)piperidine-1-carboxamide