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1-ethyl-3-(piperidine-1-carbonyl)-N-(quinolin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
8-(5-cyano-4,6-dimethylpyridin-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
8-methoxy-4-methyl-2-(1H-pyrazol-3-yl)quinoline
N-(2-hydroxyethyl)-N-methyl-1-[1-(naphthalen-2-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-N-(pyridin-2-ylmethyl)acetamide
(1S,3R)-3-amino-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}cyclopentane-1-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(morpholin-4-yl)ethyl]acetamide
1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-4-carboxamide
2,5-dimethyl-3-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[(6-methylpyridin-2-yl)methyl]amine
2-(3-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
1,9-dimethyl-4-{[4-(trifluoromethyl)phenyl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[1-(2,3-dihydro-1H-indene-1-carbonyl)azetidin-3-yl]pyridine
5-{[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-methyl-1,3-thiazole
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(3-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
5-(1-cyclobutylpyrrolidin-2-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}thiophene-2-carboxamide
6-[2-(4-fluorophenyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl(2-phenylethyl){[3-(pyrrolidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}amine
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-(piperidin-1-yl)acetamide
3-benzyl-4-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperazin-2-one
N-methyl-4-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H-imidazol-2-yl}benzene-1-sulfonamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-(prop-2-en-1-yloxy)benzamide
(1S,5R)-3-(5-chloropyridin-2-yl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-methyl-6-{4-[(3-methyl-1-benzothiophen-2-yl)methyl]piperazin-1-yl}pyrimidin-2-amine
N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-(thiophen-3-yl)acetamide
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-(1H-pyrazol-1-yl)pyrimidine
2-(4-ethyl-1,3-thiazol-2-yl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(3-fluorophenyl)-5-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
N-(2-hydroxyethyl)-1-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
1-ethyl-N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-3-methyl-1H-pyrazole-4-carboxamide
N-(propan-2-yl)-2-{1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
4-({4-methyl-5-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-methyl-4-(4-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}phenyl)butan-2-ol
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[methyl(2-methylpropyl)amino]methyl}piperidin-2-one
N-(1-cycloheptylpiperidin-3-yl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
3-[(tert-butylamino)methyl]-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
1-[1-(pyrimidin-2-yl)piperidin-4-yl]azepane
3-{4-[5-(morpholin-4-ylmethyl)pyridin-2-yl]phenyl}propanoic acid
methyl (2S,4R)-1-methyl-4-{2-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}pyrrolidine-2-carboxylate
(1R,5S)-6-[(2-butoxy-3-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-[4-(1-ethoxyethyl)phenyl]-1,2-dihydropyridin-2-one
4-(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)thiomorpholine
(5S)-5-({[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl](pyridin-3-ylmethyl)amino}methyl)pyrrolidin-2-one
1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
1-[(2-methyl-1,3-thiazol-5-yl)methyl]-3-[4-(trifluoromethyl)benzoyl]piperidine
ethyl 1-[2-(2-oxopyrrolidin-1-yl)ethyl]-1H-imidazole-2-carboxylate
N-(1,3-dihydroxypropan-2-yl)-5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-4-(piperidin-3-yl)benzamide