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N,N-dimethyl-3-[3-(1H-pyrazol-3-yl)phenyl]benzamide
2-(3-methoxyphenoxymethyl)-N-(2-methylprop-2-en-1-yl)-1,3-oxazole-4-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-5-hydroxy-N-(2-methoxyethyl)pyridine-2-carboxamide
3-chloro-4-({1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
N-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]-4-(pyrrolidin-1-ylmethyl)benzamide
3-(3-fluorophenyl)-3-{2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]acetamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 1-(2,2-dimethylpropanoyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
4-fluoro-N-(3-{4-[(pyridin-4-ylmethyl)amino]piperidin-1-yl}phenyl)benzene-1-sulfonamide
2-(adamantan-1-yl)-4-hydroxy-N-(2-hydroxypropyl)pyrimidine-5-carboxamide
ethyl 3-[(2-fluorophenyl)methyl]-1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidine-3-carboxylate
4-{4-[1-(3-chloro-4-fluorophenyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine
1-{2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
(1R,5R)-3-(pyridine-2-carbonyl)-6-(1,3-thiazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-(1-phenyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(furan-2-ylmethyl)-4-[2-(2-phenylethynyl)phenyl]-1H-1,2,3-triazole
2-({4-[4-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)pyridine
1-[(2-fluorophenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
methyl (2S,4R)-4-(5-chloro-3-methyl-1H-indole-2-amido)-1-[(3-ethoxy-4-hydroxyphenyl)methyl]pyrrolidine-2-carboxylate
4-[2-(difluoromethoxy)benzoyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-(4-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}phenyl)acetamide
3-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]urea
4-(2-methylphenyl)-N-(1,3,4-thiadiazol-2-yl)-1,4-diazepane-1-carboxamide
2-(pyridin-2-ylmethyl)-9-[4-(pyrrolidin-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(3S)-4-(3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanoyl)-1,3-dimethylpiperazin-2-one
N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)oxan-4-amine
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(4-phenylbenzoyl)-1,4-diazepan-5-one
2-(4-methoxyphenyl)-5-{[4-(pyrimidin-4-yl)piperidin-1-yl]methyl}pyrimidine
1-(4-{2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}piperidin-1-yl)ethan-1-one
N-ethyl-4-hydroxy-2-(3-methylphenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidine-5-carboxamide
(1s,4s)-4-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-ylmethyl}cyclohexan-1-amine
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-imidazol-1-yl)propan-1-one
1-({4-methyl-5-[1-(6-methylpyrimidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
N-cyclopropyl-1-(2-{1-[2-(3-methylphenyl)acetyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-(morpholin-2-yl)acetamide
1-(3-chloro-2-fluorophenyl)-3-methyl-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazole
2-[4-(5-chloro-2,3-dihydro-1H-indole-2-carbonyl)-1,4-diazepan-1-yl]-N,N-dimethylacetamide
4-(2-phenoxyacetyl)-N-[4-(propan-2-yl)phenyl]piperazine-1-carboxamide
5-{1-[2-(5-phenyl-4H-1,2,4-triazol-3-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)-2-(pyridin-4-yl)acetamide
2-{5-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-indole
3-fluoro-5-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]benzonitrile
1-(4-methylpiperidin-1-yl)-3-{[1-(2-methylpropyl)piperidin-4-yl]amino}propan-1-one
4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-(1,2,5-thiadiazole-3-carbonyl)piperidine
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[2-(4-methylphenyl)ethyl]amine
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N,N-dimethylpyridine-3-carboxamide
1-(3,4-dimethylphenyl)-3-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}urea
2-{2-methyl-4-[3-(1H-pyrazol-3-yl)phenyl]phenoxy}acetamide
3-{[1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidin-4-yl]oxy}pyridine