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4-[(1-benzyl-1H-imidazol-2-yl)methyl]-3-butyl-1-methylpiperazin-2-one
N-cyclohexyl-4-[3-(1-methyl-1H-pyrazol-4-yl)propanamido]piperidine-1-carboxamide
1-ethyl-4-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
7-[2-(4-chlorophenyl)-2-hydroxyacetyl]-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(oxolan-2-ylmethyl)-8-(pyridine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}azepane-4-carboxamide
(2S,4R)-4-amino-1-(3-cyclopentaneamido-4-methylbenzoyl)-N-ethylpyrrolidine-2-carboxamide
7-fluoro-N,3-dimethyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1H-indole-2-carboxamide
3-[5-(1-benzofuran-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]benzonitrile
8-chloro-4-[4-(4-methoxybutyl)piperazine-1-carbonyl]-2-methylquinoline
1-butyl-3-(2-methyl-1,3-thiazol-4-yl)-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazole
2-[2-(3-cyanophenyl)-1H-imidazol-1-yl]-N-(2,3,4-trifluorophenyl)acetamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-(2-phenylethyl)-N-(propan-2-yl)acetamide
methyl[(5-methylthiophen-2-yl)methyl]{[5-(pyridin-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amine
2-(4-chlorophenyl)-4-[4-(morpholine-4-carbonyl)pyridin-2-yl]morpholine
2-{[2-(1-benzofuran-5-yl)-1H-imidazol-1-yl]methyl}-3-methylpyridine
1-methyl-5-[(2-methylpropyl)amino]-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{2-oxo-2-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethyl}methanesulfonamide
N3-butyl-1-cyclohexyl-4-oxo-N5-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanol
1-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]-1,2-dihydroquinoxalin-2-one
2-(dimethylamino)-N,4-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]pyrimidine-5-carboxamide
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
8-[(4-ethoxyphenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
(3aR,6aR)-2-acetyl-N-[4-(pyridin-2-yl)butyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-[(4-chlorophenyl)methyl]-N-(1-methoxybutan-2-yl)-1,3-benzoxazole-5-carboxamide
4-(2,4-dimethyl-1,4-diazepane-1-carbonyl)-2-(1-ethyl-1H-pyrazol-4-yl)-6-fluoroquinoline
N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
2-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}-6-methylpyridine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]propane-2-sulfonamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[(3S)-3-fluoropyrrolidin-1-yl]ethan-1-one
(3aS,6aS)-1-methyl-5-{2-methylthieno[2,3-d]pyrimidin-4-yl}-octahydropyrrolo[3,4-b]pyrrole
N-(1-benzothiophen-2-ylmethyl)-N-methyl-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]acetamide
2-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
2-[5-(2,3-dihydro-1-benzothiophen-2-yl)-3-(4-fluorophenoxymethyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-methyl-4-[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]-1,4-diazepane
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-1H-pyrazole-3-carboxamide
N-cyclopropyl-1-[1-(2-ethylpyridine-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}-N-[2-(pyridin-4-yl)ethyl]benzamide
benzyl(ethyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
1-({4-methyl-5-[1-(pyridine-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
2-methyl-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-(3-hydroxyphenyl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-oxopyrrolidine-3-carboxamide
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-(3-methyl-2-oxoimidazolidin-1-yl)acetamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-4-phenylbutane-1,4-dione
(1S,5R)-6-(2-methoxyethyl)-3-{2-[(3-methoxyphenyl)sulfanyl]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-{[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one