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N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-2-(1H-1,2,4-triazol-1-yl)acetamide
N-(1-methanesulfonylpiperidin-4-yl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methanol
1-cyclopropyl-4-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]pyrrolidin-2-one
2-{[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]amino}-N,N-dimethylpyridine-3-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}acetamide
7-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
4-[1-benzyl-5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
(2S,4S)-N-ethyl-4-(furan-2-amido)-1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]pyrrolidine-2-carboxamide
3-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}-1-(4-ethylpiperazin-1-yl)propan-1-one
N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]-2H-1,3-benzodioxole-5-carboxamide
{1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-3-(2-phenoxyethyl)piperidin-3-yl}methanol
1-({3-[(dimethyl-1,2-oxazol-4-yl)carbamoyl]phenyl}methyl)-N-ethylpyrrolidine-3-carboxamide
N-butyl-N-[(2-fluorophenyl)methyl]-2-(1,2,3,6-tetrahydropyridin-4-yl)acetamide
N-[3-(1H-indazol-1-yl)propyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
N-benzyl-N-methyl-3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)acetamide
(3S)-3-({[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}amino)azepan-2-one
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-[(3-methylpyridin-4-yl)methyl]propanamide
[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl](methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-4-(4-methylphenoxy)piperidine-4-carboxamide
1-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)-4-methylpiperazine
(1S,5R)-6-(cyclobutylmethyl)-3-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2,6-difluoro-4-methoxy-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
1-{2-hydroxy-3-[2-methoxy-4-(morpholin-4-ylmethyl)phenoxy]propyl}piperidin-4-ol
(1r,4r)-4-{[6-amino-2-(benzylsulfanyl)pyrimidin-4-yl]amino}cyclohexan-1-ol
[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(furan-2-yl)ethane-1,2-dione
N-[(2S,4R,6S)-2-(3-cyclohexyl-1H-pyrazol-4-yl)-6-(2-methylpropyl)oxan-4-yl]acetamide
1-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-2-methyl-1-benzofuran-5-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(3-hydroxypropyl)-N-(pyridin-4-ylmethyl)propanamide
1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-3-({[1-(thiophen-2-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
N3-({2-[(dimethylamino)methyl]phenyl}methyl)-N1,N1,N3-trimethylpiperidine-1,3-dicarboxamide
2-(2-chlorophenyl)-3-methyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
5-amino-4-chloro-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1H-pyrazole-3-carboxamide
5-{[2-(1H-imidazol-4-yl)ethyl]carbamoyl}-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-4-(morpholin-4-yl)benzamide
2-(4-fluorophenyl)-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
(4aR,8aS)-6-(2H-1,3-benzodioxol-5-ylmethyl)-1-[3-(morpholin-4-yl)propyl]-decahydro-1,6-naphthyridin-2-one
N-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-2-[4-(3-methoxypyrazin-2-yl)-1H-pyrazol-1-yl]acetamide
cyclohexyl({4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl})methanol
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[(1r,4r)-4-hydroxycyclohexyl]acetamide
N-{1-[1-(3-fluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
1-(furan-2-yl)-2-[3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]ethane-1,2-dione
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1-[2-(1H-pyrazol-1-yl)phenyl]urea
2-(carbamoylamino)-N-[2-(4-cycloheptylmorpholin-2-yl)ethyl]acetamide
4-[(1-hydroxy-3-methylbutan-2-yl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid