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N-[2-(furan-2-yl)ethyl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-[(5-ethylpyridin-2-yl)methyl]-N-methylthian-4-amine
N-[1-(2-methoxyphenoxy)propan-2-yl]-1-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
4-hydroxy-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
[(3R,4R)-1-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[(3R,4R)-3-hydroxy-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-1-yl]pent-4-en-1-one
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)-2-(4-oxo-1,4-dihydroquinolin-1-yl)acetamide
N-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-(pyridin-2-ylmethyl)piperidin-3-amine
[(1-ethyl-1H-imidazol-2-yl)methyl]({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
3-[(1-acetylpiperidin-4-yl)oxy]-N-(cyclohex-1-en-1-ylmethyl)-4-methoxybenzamide
1-[2-chloro-5-(piperidine-1-carbonyl)phenyl]-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
N-[(5-methylthiophen-2-yl)methyl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
1-[(5-ethylpyridin-2-yl)methyl]-1-methyl-3-[2-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
5-{2-oxo-2-[4-(2-phenylethyl)piperidin-1-yl]ethyl}-3-propylimidazolidine-2,4-dione
(2S,4S)-N-ethyl-4-(furan-3-amido)-1-[2-(thiophen-3-yl)acetyl]pyrrolidine-2-carboxamide
4-{1-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]azetidin-3-yl}pyridine
(1s,4s)-N-[(2,4-dimethoxyphenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexan-1-amine
2-{[3-(hydroxymethyl)-3-methylpiperidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
7-[2-(2-ethylphenoxy)ethyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
7-{[(3-hydroxy-3-methylbutyl)(methyl)amino]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
1-[1-(methoxymethyl)cyclobutanecarbonyl]-3-(3-methoxyphenoxymethyl)piperidine
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
5-(2-chloro-4-fluorophenoxymethyl)-N-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-1,2-oxazole-3-carboxamide
1-benzoyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]piperidin-4-amine
methyl 5-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-methyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1H-indole-6-carboxamide
(4aS,7aR)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-(1H-1,2,3,4-tetrazol-5-yl)ethan-1-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
(2R,3R,6R)-3-(4-methylphenyl)-5-(1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{2-oxo-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]ethyl}-3,4-dihydro-1,2,3-benzotriazin-4-one
1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-(methylamino)-2-phenylethan-1-one
1-(2-methyl-1,3-thiazole-5-carbonyl)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-ethyl-N-(3-methylbutyl)-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](methyl){[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
7-(5,6-dimethylpyrimidin-4-yl)-N,N,2-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}cyclobutanecarboxamide
({5-methanesulfonyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
[(3S,5R)-5-[(dimethylamino)methyl]-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl]methanol
butyl[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](furan-2-ylmethyl)amine
2-[2,4-dichloro-3-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-4-carbonitrile
(3S,4R)-1-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
3,5-difluoro-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}pyridine-2-carboxamide
N-{[7-(4-chlorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
2-amino-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)-4-[3-(1H-pyrazol-1-yl)phenyl]pyridine-3-carbonitrile
5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]-4-[1-(1,3-thiazole-5-carbonyl)piperidin-3-yl]pyrimidine
(3S,4S)-1-[4-(1H-imidazol-1-yl)benzoyl]-4-propylpyrrolidine-3-carboxylic acid
2-methoxy-5-({[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amino}methyl)phenol