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1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-3-carboxamide
5-[(5-methylthiophen-2-yl)sulfonyl]-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
5-{3-[2-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}quinoxaline
6-methyl-2-oxo-5-({3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}carbonyl)-1,2-dihydropyridine-3-carbonitrile
5-[1-(4-fluorophenyl)cyclopropyl]-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
ethyl 1-[5-(benzylcarbamoyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carbonyl]piperidine-3-carboxylate
N-[4-oxo-4-(3-oxo-4-phenylpiperazin-1-yl)butyl]acetamide
5-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]-3-chloro-1,2-dihydropyridin-2-one
N-(3-hydroxypropyl)-N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
1-({5-[1-(2-methoxyethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
4-(5-ethoxyfuran-2-amido)-N-ethylpiperidine-1-carboxamide
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[4-(1-methyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]acetamide
1-(2-methoxyacetyl)-N,4-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}piperazine-2-carboxamide
4-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperazine-1-sulfonamide
4-methyl-6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-phenylpyrimidine
3-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-[5-(5-ethyl-1,3,4-oxadiazol-2-yl)-2-methoxyphenyl]urea
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-[1-(pyridin-4-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
3-[3-(furan-2-yl)phenyl]-1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1-methylurea
6-(4-methoxyphenyl)-7-(prop-2-en-1-yl)-2-(pyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
4-({[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amino}methyl)-2,6-dimethylphenol
1-[(2,4-dimethoxyphenyl)methyl]-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
[(2,3-difluorophenyl)methyl]({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})amine
(2R,3R,6R)-3-(4-fluorophenyl)-5-(2-methylfuran-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2-methylphenyl)-2-{4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}acetamide
1-(2-methylpropanoyl)-4-(2-phenylethyl)piperidine-4-carboxylic acid
N-ethyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
3-(2-methylphenyl)-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-3-phenylpropan-1-one
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
1-{5-[3-(2-phenylethyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
4-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}-1-(propan-2-yl)pyrrolidin-2-one
1-benzyl-N,N-dimethyl-5-{[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(3-chlorophenyl)-4-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]piperazine
1-(2,3-dihydro-1H-indol-1-yl)-2-{2-oxa-7-azaspiro[4.5]decan-7-yl}ethan-1-one
1-[1-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidin-4-yl]ethan-1-ol
N-({7-[(3-ethoxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
2-(5-fluoroquinolin-8-yl)-N-methylpyridine-4-carboxamide
6-(pyridin-4-yl)-2-[4-(thiomorpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
1-(furan-3-ylmethyl)-3-[4-(methylsulfanyl)benzoyl]piperidine
N-[2-(azepan-1-yl)ethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-(propan-2-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
2-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-1-(pyridin-4-yl)ethan-1-ol
3-methyl-4-oxo-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-3,4-dihydroquinazoline-7-carboxamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-[5-(propan-2-yl)pyrimidin-4-yl]pyrrolidin-3-amine
2-cyclopropyl-4-phenyl-9-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-(benzyloxy)-1-cyclohexyl-4-[5-(methoxymethyl)furan-2-carbonyl]-1,4-diazepan-2-one
3-[1-(4-methanesulfonylbenzoyl)piperidin-3-yl]benzoic acid
2,6-dimethyl-N-[(3R,4S)-1-[(methylcarbamoyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]pyrimidine-4-carboxamide
(4aS,7aR)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(pyridin-3-yl)piperidin-4-ol