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N-(3,4-dimethylphenyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-amine
3-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-1-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]urea
(3aR,5S,6S,7aS)-2-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]-octahydro-1H-isoindole-5,6-diol
4-[(4-fluorophenyl)methyl]-9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-8-methoxyquinoline
{4-methyl-5-[(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-4-yl)methyl]-4H-1,2,4-triazol-3-yl}methanol
2-methyl-8-[(E)-2-phenylethenesulfonyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[3-oxo-9-(quinolin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
2-[(2-amino-6-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}pyrimidin-4-yl)amino]ethan-1-ol
2-(3,5-dimethyl-4-{[(pyridin-3-yl)carbamoyl]amino}-1H-pyrazol-1-yl)acetic acid
3-[2-(4-fluorophenyl)ethyl]-1-(oxane-4-carbonyl)piperidine
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]pyridine-4-carboxamide
3-[2-(benzyloxy)phenyl]-1-[3-(morpholin-4-yl)propyl]urea
N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
3-(4-chlorophenyl)-5-cyclobutanecarbonyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
dimethyl({5-[(4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazin-1-yl)methyl]thiophen-3-yl}methyl)amine
methyl 2-[1-(3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-3-oxopiperazin-2-yl]acetate
2-amino-4-(3,5-dimethyl-1H-pyrazol-4-yl)-6-(4-hydroxyphenyl)-5-methylpyridine-3-carbonitrile
2-[4-(1H-imidazol-4-ylmethyl)morpholin-3-yl]-N-[2-(methylsulfanyl)phenyl]acetamide
methyl 4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-5-methylthieno[2,3-d]pyrimidine-6-carboxylate
5-chloro-N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}quinoline
(1S,5R)-6-benzyl-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-1-(furan-2-ylmethyl)piperidine-3-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-(hydroxymethyl)cyclopropane-1-carboxamide
(2S)-2-amino-N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)hexanamide
2-(4-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}phenoxy)acetic acid
4-[(diethylamino)methyl]-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-ethylfuran-2-carboxamide
6-(2,5-dimethylfuran-3-yl)-2-[(3R)-3-hydroxypyrrolidine-1-carbonyl]-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-{2-[4-(pyrrolidin-1-yl)piperidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
(1S,3R)-3-amino-N-{[3-(3-methylbutyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentane-1-carboxamide
2-amino-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)-4-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]pyridine-3-carbonitrile
6-[(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)amino]pyridine-3-carboxamide
1-(oxane-4-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
ethyl 3-benzyl-1-(3-phenylprop-2-ynoyl)piperidine-3-carboxylate
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-3-propylpiperidin-3-yl)methanol
N-methyl-3-(1H-pyrazol-1-ylmethyl)-N-[1-(pyrimidin-4-yl)ethyl]benzamide
6-(2-fluorophenyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2,4-difluoro-3-methoxy-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)benzamide
2-(ethoxymethyl)-N-(furan-3-ylmethyl)-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(4aS,8aR)-6-[2-(dimethylamino)acetyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-[(2,5-dioxopyrrolidin-3-yl)sulfanyl]-N-(furan-2-ylmethyl)benzamide
4-[4-(4-methylpiperazin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide