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N-[2-(2-methylpropanesulfonyl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
2,3-dimethyl-4-oxo-N-[2-(propan-2-yl)phenyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
(2E)-N-({3-methyl-7-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenylprop-2-enamide
methyl 3-{imidazo[1,2-a]pyridine-2-carbonyl}-9-[2-(1-methylpyrrolidin-2-yl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[3-(4-{[3-(1H-1,2,3-benzotriazol-1-yl)propyl]amino}piperidin-1-yl)phenyl]ethane-1-sulfonamide
8-[(1-benzyl-1H-imidazol-5-yl)methyl]-8-azaspiro[4.5]decane-7,9-dione
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-2-{[6-(pyrrolidin-1-yl)pyridazin-3-yl]oxy}acetamide
2-{4-[1-(1H-imidazole-5-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
(2E)-N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-3-(thiophen-2-yl)prop-2-enamide
2-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-5-methylpyrazine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
[(3R,4R)-1-(naphthalen-2-ylmethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-(3-methylthiophen-2-yl)-4-phenyl-1H-imidazole
(1R,2R,3S,4S)-3-amino-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}bicyclo[2.2.1]heptane-2-carboxamide
4-[1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)piperidine-4-carbonyl]morpholine
(3aR,6aR)-2-(2-hydroxyethyl)-5-[1-(methoxymethyl)cyclobutanecarbonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1R,2S)-2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)cyclopentan-1-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[methyl(thian-4-yl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-({[(1-cyclopropyl-1H-imidazol-5-yl)methyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
ethyl 1-cyclopentyl-4-(3-phenylpropyl)piperidine-4-carboxylate
(4aS,8aR)-1-(4-hydroxybutyl)-6-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-decahydro-1,6-naphthyridin-2-one
(3aR,6aS)-5-(2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1S,5R)-3-(6-aminopyridine-3-carbonyl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(but-2-yn-1-yl)-5-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione
N-ethyl-3-(4-phenylbenzoyl)piperidine-1-carboxamide
2-benzyl-8-(3-fluoropyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(2-carboxyphenyl)methyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
8-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
4-(1H-imidazol-1-ylmethyl)-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
(5S,9aS,9bS)-2-(3-methoxyphenyl)-5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-methyl-2-{2-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,3-benzodiazole
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-(2-oxopiperidin-1-yl)acetamide
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-4-yl)ethyl]acetamide
1-methyl-4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(3-fluorophenyl)methyl]-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
(1s,4s)-4-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}cyclohexan-1-amine
3-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]piperidin-2-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
{5-methyl-3-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-oxazol-4-yl}methanol
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl](oxolan-2-ylmethyl)amine
1-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
4-benzyl-1-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]pyrrolidin-2-one
(3R,4R)-4-amino-1-{1-[(4-phenylphenyl)methyl]-1H-1,2,3,4-tetrazol-5-yl}piperidin-3-ol
3-[1-(2,3-dimethoxybenzoyl)piperidin-3-yl]-N-(4-fluoro-2-methylphenyl)propanamide
2,4-dimethyl-N-[1-(4-{[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]benzamide
1-[(2-phenyl-1,3-oxazol-4-yl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
7-[3-(pyridin-3-yloxy)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
4-[4-(ethylsulfanyl)phenyl]-6-methylpyrimidin-2-amine
1-(2-methoxyphenyl)-3-(1-{1-[2-(3-methylphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
{4-[(3-fluorophenyl)methyl]-1-(4-methylpyrimidin-2-yl)piperidin-4-yl}methanol