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1-(1,2,3,4-tetrahydroisoquinolin-2-yl)-3-[4-({[2-(1,3-thiazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methylpiperazine
3-(1,3-benzothiazol-2-yl)-N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}propanamide
[5-({4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)furan-2-yl]methanol
3-(6-fluoroquinolin-8-yl)-N-methylpyrazin-2-amine
3-({[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)-2,2-dimethylpropan-1-ol
2-{1-[(6-methylpyridin-2-yl)methyl]-4-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperazin-2-yl}ethan-1-ol
3-(3-methoxybenzoyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
2-ethyl-8-[(1-ethyl-1H-imidazol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperidin-4-amine
6-[3-(3-fluorophenyl)benzoyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
(4aS,8aR)-6-[3-(2,4-difluorophenyl)propanoyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
4-{[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
3-{[(1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl)oxy]methyl}pyridine
3-(6-methoxypyridazin-3-yl)quinoline
2-(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)ethan-1-amine
(2S)-2-hydroxy-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-2-phenylacetamide
N-ethyl-6-(3-methoxypiperidin-1-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)-5-(methoxymethyl)furan-2-carboxamide
1-[4-(2,5-dimethylphenyl)piperazin-1-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
2-[(1R,2S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecan-11-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
1-[1-(2-hydroxybutyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-[(2-fluorophenyl)formamido]-N-(1-methoxypropan-2-yl)propanamide
({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)(oxolan-3-ylmethyl)amine
N-methyl-N-(2-methylpropyl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N,2,6-trimethyl-N-[1-(pyridin-4-yl)ethyl]pyrimidine-4-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-[methyl(1-methylpiperidin-4-yl)amino]acetamide
4-({4-methyl-5-[1-(pyrimidin-2-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
ethyl 4-({2,7-diazaspiro[4.5]decane-2-carbonyl}amino)benzoate
6-oxo-N-[2-(1,3-thiazol-4-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
4,6-dimethyl-2-oxo-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-1,2-dihydropyridine-3-carboxamide
2-benzamido-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
N-(3-methoxypropyl)-N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
1-[4-methyl-2-(3-phenylpiperazin-1-yl)pyrimidin-5-yl]ethan-1-one
(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(3-hydroxy-2,2-dimethylpropyl)(methyl)amino]methyl}piperidin-2-one
1-(1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}azetidin-3-yl)-3,5-dimethyl-1H-pyrazole
(4aR,7aS)-1-methyl-4-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(cyclopropylmethyl)-1-(2-hydroxyethyl)-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
(3S,9aR)-3-benzyl-2-methyl-8-(4-methylbenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{1-[7-(1-cyclobutylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-2-(dimethylamino)acetamide
N-methyl-2-(pyridin-4-yl)-N-(quinolin-5-ylmethyl)pyrimidine-5-carboxamide
5-(propan-2-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-(2-hydroxyphenyl)ethan-1-one
(2E)-3-(1,3-benzothiazol-2-yl)-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methylprop-2-enamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(2-oxoazepan-1-yl)propanamide
methyl 6-[(2-fluoro-4-methoxyphenyl)methyl]-2-[(3-methylbutyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(3-cyano-4-methylphenyl)-4-[2-(methylsulfanyl)ethyl]piperazine-1-carboxamide