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1-(2-ethoxyethyl)-N-(1H-indol-2-ylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-[4-(2-methylpropyl)piperazin-1-yl]-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
5-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-2-(pyridin-2-yl)pyrimidine
2-{4-[(2,3-difluorophenyl)methyl]-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
4-{1-[1-(benzenesulfonyl)piperidin-4-yl]-1H-imidazol-2-yl}pyridine
2-methoxy-2-methyl-1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
1-[(2,5-difluorophenyl)methyl]-4-[2-(4-methyl-1,4-diazepane-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
1-methyl-4-[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-1,4-diazepane
[benzyl(methyl)sulfamoyl]({4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl})amine
4-{[(2-methoxyethyl)[(4-methylphenyl)methyl]amino]methyl}-N-methylbenzene-1-sulfonamide
3-{[4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]methyl}-1H-indole
4-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}benzoic acid
5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-(3-methoxyphenyl)-1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidine
6-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyethyl)pyrrolidin-3-yl]-3-(methylsulfanyl)propanamide
6-(2-fluoro-4-methoxyphenyl)-N-(2-hydroxyethyl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(2S,4R)-4-amino-1-{2,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carbonyl}-N-ethylpyrrolidine-2-carboxamide
N-(2-{5-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}ethyl)acetamide
4,4,4-trifluoro-N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}butanamide
1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyridin-2-ylmethyl)-1,4-diazepane
3-hydroxy-3-({[(5-methylfuran-2-yl)methyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one
(2R)-2-cyclohexyl-2-hydroxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
4-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,3-thiadiazole
1-{[4-(benzyloxy)phenyl]methyl}-N-ethylpyrrolidine-3-carboxamide
1-(2-{2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
4-cyclopentyl-3-(3-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-(4-methoxy-2-methylbenzoyl)piperidine
2-(dimethylamino)-7-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(4-fluorophenyl)methyl]-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(propan-2-yl)-1,4-diazepane
N-methyl-N-[(4-phenoxyphenyl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-3-(4-methylpiperazin-1-yl)propan-1-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(methylsulfanyl)ethan-1-one
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)thiophene-3-carboxamide
2-cyclopropyl-5-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-3,4-dihydropyrimidin-4-one
N-[(3R,4S)-4-propyl-1-[2-(2H-1,2,3-triazol-2-yl)acetyl]pyrrolidin-3-yl]methanesulfonamide
N-[(2R,3R)-2-(pyridin-4-ylmethoxy)-1'-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
3-({[5-(hydroxymethyl)furan-2-yl]methyl}amino)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-5-[(propan-2-yl)sulfamoyl]benzamide
N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
N-[4-(4-{[3-(4-methyl-1,3-thiazol-5-yl)propyl]amino}piperidin-1-yl)phenyl]benzenesulfonamide
2-(4-fluorophenyl)-1-{4-[3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}ethan-1-one
N-({7-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
1-methyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)piperidine-4-carboxamide
[3-(cyclopropylmethyl)-1-[(2-ethyl-1,3-thiazol-4-yl)methyl]piperidin-3-yl]methanol
5-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
(4aR,7aS)-1-(cyclopropylmethyl)-4-{[3-(2-hydroxyethoxy)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,3-dimethoxy-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)benzamide
N-cyclopentyl-2-cyclopropyl-N-[(2,4-dimethoxyphenyl)methyl]pyrimidine-5-carboxamide