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2-[(3S,4R)-4-amino-1-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}pyrrolidin-3-yl]ethan-1-ol
1-[(4-fluorophenyl)methyl]-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-methyl-N-[(1-phenyl-1H-pyrazol-5-yl)methyl]-N-(pyridin-4-ylmethyl)piperidin-4-amine
5-(1H-indol-1-ylmethyl)-N-[(3-methylpyridin-4-yl)methyl]-1H-pyrazole-3-carboxamide
(1R,5S,6R)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(quinolin-4-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
(4aS,7aR)-1-[(3-hydroxyphenyl)methyl]-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2R,3R)-1'-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
4-{[3-(trifluoromethyl)-1H-pyrazol-5-yl]methyl}-1,4-oxazepane
(3R,9aR)-3-methyl-8-(3-phenylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-cyclopentyl-5-[(4-acetamidophenyl)methyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[(4-ethylpiperazin-1-yl)methyl]-N-(furan-2-ylmethyl)-N-methyl-1,2-oxazole-3-carboxamide
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxypropan-1-one
3-{3-[5-benzoyl-3-(piperidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-1-yl]propyl}pyridine
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidine
(2R,3S,6R)-5-(ethanesulfonyl)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
5-(5-propylthiophene-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydrophthalazin-1-one
N-ethyl-N-(2-hydroxyethyl)-5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
1-(4-tert-butylphenyl)-3-[(5-methyl-1H-imidazol-4-yl)methyl]urea
5-[2-(methoxymethyl)piperidine-1-carbonyl]-2-(2-phenylethyl)-1,3-benzoxazole
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
4-{1-[(5-chlorothiophen-2-yl)sulfonyl]piperidin-4-yl}-5-[3-(trifluoromethyl)phenyl]pyrimidine
5-chloro-N-[2-(1-ethylpiperidin-3-yl)ethyl]-1,3-dimethyl-1H-pyrazole-4-sulfonamide
4-{4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]piperidine-1-carbonyl}pyridin-2-amine
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
N-(2,3-dihydro-1H-inden-2-yl)-1-methyl-1H-pyrazole-5-carboxamide
N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carboxamide
1-[1-(1-ethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-(phenylamino)pyrimidine-5-carboxamide
5-[4-(aminomethyl)piperidin-1-yl]-2-[(1-benzyl-1H-imidazol-2-yl)methyl]-2,3-dihydropyridazin-3-one
3-[3-methyl-1-(2-methylphenyl)-1H-pyrazol-5-yl]-1-(1,4-oxazepan-6-ylmethyl)urea
2-(4-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-1,3-benzoxazole
methyl 4-{[3-(carbamoylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}benzoate
1-[4-(pyridin-2-yl)piperazin-1-yl]-3-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}propan-1-one
2-methyl-2-(methylamino)-1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
4-(6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrazine-2-carbonyl)morpholine
3,5-dimethyl-4-[1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]-1,2-oxazole
5-[1-(2,3-dihydro-1H-inden-2-yl)-1H-pyrazol-3-yl]-4-methyl-N-[(3,4,5-trimethoxyphenyl)methyl]-1,3-thiazol-2-amine
2-[4-phenyl-5-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]acetic acid
1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyridin-2-yl)piperazine
1-{1-[(2,4-dimethoxyphenyl)methyl]-4-phenylpiperidin-4-yl}ethan-1-one
1-(5-fluoro-2-methylbenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N1-(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)propane-1,3-diamine
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-2-yl)ethyl]acetamide
2-cyclopropyl-8-{[4-(difluoromethoxy)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
N-{[1-(3,5-dimethylphenyl)cyclopentyl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide