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2-methyl-6-(3-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
5-(1-butyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)-1H-indole
N-butyl-1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-cycloheptyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
3-[(2-methylpyrrolidin-1-yl)methyl]-N-(1-oxo-2,3-dihydro-1H-inden-5-yl)benzamide
1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(2,2-dimethyloxan-4-yl)-1H-1,2,3-triazole
4-(2-{2-[4-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}propyl)pyridine
methyl (2S,4R)-4-[(3-chlorophenyl)methanesulfonamido]-1-methylpyrrolidine-2-carboxylate
4-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-methyl-4-oxobutanamide
1-{[1-(3-methylpyridin-4-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
methyl 8-{[2-(furan-2-yl)phenyl]methyl}-1-methoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
(2S,4S)-N-[(4-methylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
{4-[(4-chlorophenyl)methyl]-1-[(2,4-dimethoxy-3-methylphenyl)methyl]piperidin-4-yl}methanol
(1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-yl)methanamine
3-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetamido]-3-phenylpropanoic acid
8-[(4-hydroxyphenyl)methyl]-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N5-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N6-(2-methoxyethyl)-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-[3-(pyridin-4-yl)-5-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-{[7-(2,6-dimethoxybenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-methylbutanamide
3-{[(2S,5R)-5-{[methyl(1-methylpiperidin-4-yl)amino]methyl}oxolan-2-yl]methyl}phenol
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-(3-phenylpropyl)-1,4-diazepane
N-methyl-2-oxo-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]piperidine-3-carboxylic acid
(2-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}phenyl)methanol
3-[2-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl]pyridine
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(diethylamino)methyl]phenoxy]-N-(3-fluorophenyl)acetamide
5-(2-chlorophenyl)-N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]furan-2-carboxamide
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(piperidine-1-carbonyl)pyridine
9-(5-propyl-1,3,4-thiadiazol-2-yl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-(5-chloropyridin-2-yl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[(1,4-dioxan-2-ylmethyl)(methyl)amino]-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-6-[4-(methylsulfanyl)phenyl]pyridine-3-carboxamide
4-{5-[2-(2-methyl-1H-imidazol-1-yl)propyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl}pyridine
N-[(5-ethylpyridin-2-yl)methyl]-N,2,8-trimethylquinoline-4-carboxamide
2-(3,4-dichlorophenyl)-4-(2-methylbenzoyl)morpholine
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(1-propyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidin-3-yl]methanol
3-(1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-N,N-dimethylpropanamide
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(3-methylpyridin-2-yl)piperazine
9-(3-hydroxybenzoyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 3-{[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]carbamoyl}benzoate
1-(azocan-1-yl)-3-[2-methoxy-4-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-{3-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]phenyl}imidazolidin-2-one
2-[(4-methoxyphenyl)methyl]-N-[3-(methylsulfanyl)propyl]-1,3-benzoxazole-6-carboxamide
N-[3-({[2-(2-oxoimidazolidin-1-yl)ethyl]carbamoyl}methoxy)phenyl]propanamide
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-fluorophenyl)urea
3-cyclopentyl-1-(4-sulfamoylphenyl)-3-(thiophen-3-ylmethyl)urea
8-(morpholine-4-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-({1-[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}methyl)pyrrolidin-2-one
N,N-diethyl-1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-4-carboxamide
4-[5-({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine