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1-cyclopropyl-N-ethyl-5-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]pyrrolidine-3-carboxamide
5-[(3S)-3-acetamidopyrrolidine-1-carbonyl]thiophene-2-carboxylic acid
({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl})amine
1-{2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-3,3-dimethylurea
4-ethyl-3-{1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(benzylamino)-1-ethyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(4-methylphenyl)-4-[2-(morpholin-4-yl)butanoyl]piperazin-2-one
3-{3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}isoquinoline
N-ethyl-N-[2-(4-methylbenzenesulfonyl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-[1-(1-methyl-1H-imidazole-5-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
2-amino-4-(2-chloro-4-hydroxy-5-methoxyphenyl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
7-[(4-fluorophenyl)methyl]-2-[3-(1H-pyrazol-4-yl)benzoyl]-2,7-diazaspiro[4.5]decane
(5-{[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]methyl}-2-(propan-2-yloxy)phenyl)methanol
3-[5-(1-methyl-1H-pyrrole-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
[4-(3-phenylpropyl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl]methanol
methyl 4-({6-hydroxy-3-oxo-4-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-1-yl}methyl)benzoate
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
[1-(2-methylquinoline-4-carbonyl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
1'-(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
4-[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]-5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidine
[(4-ethylphenyl)methyl]({[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl})methylamine
N-{3-[2-(propan-2-yloxy)phenyl]phenyl}acetamide
(1S)-3-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1-phenylpropan-1-ol
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
1-(4-hydroxyphenyl)-N-[(5-methylpyrazin-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
4-{1-[2-methoxy-2-(thiophen-2-yl)ethyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
1-(2-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-2-oxoethyl)-2-methyl-1H-indole-3-carbonitrile
1,3-dimethyl-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]-1H-pyrazole-5-carboxamide
(3R,5S)-N3-(4-fluorophenyl)-N5-[(4-methoxyphenyl)methyl]-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
1-[5-(5-fluoro-2-methylphenyl)-1H-1,2,4-triazol-1-yl]butan-2-ol
2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrazine
1-[(1-{[5-(4-methoxyphenyl)furan-2-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
8-methoxy-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
[(4-ethoxyphenyl)methyl](methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
1-[2-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)ethyl]cyclopentan-1-ol
6-methyl-4-oxo-N-(oxolan-2-ylmethyl)-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-methyl-N-[(5-methylpyrazin-2-yl)methyl]-2-(thiophen-2-ylformamido)propanamide
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl][(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]methylamine
4-({[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]amino}methyl)-2-methoxyphenol
1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
1'-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}spiro[indene-1,4'-piperidine]
3-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methoxypyridine
1-{4-[(1-ethyl-1H-indol-6-yl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
4-{4-[({1-[(3-methoxyphenyl)methyl]piperidin-3-yl}amino)methyl]phenyl}-2-methylbut-3-yn-2-ol
N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]-5-[(methylsulfanyl)methyl]furan-2-carboxamide
(4aR,8aR)-6-(3-methoxybenzoyl)-1-(3-phenylbutyl)-decahydro-1,6-naphthyridine
3-methyl-1-(2-phenylethyl)-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazole
2-{[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]amino}ethan-1-ol