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3-cyclopropyl-5-[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]-1-propyl-1H-1,2,4-triazole
4,6-dimethyl-3-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
(1H-1,3-benzodiazol-2-ylmethyl)[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]methylamine
2-{[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]methyl}-6,8-dimethyl-1,4-dihydroquinolin-4-one
2,3-dimethyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}quinoxaline-6-carboxamide
1-{[1-(4-fluorophenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}azepan-2-one
2-(4-methoxyphenyl)-5-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
2-amino-1-{6-methyl-5-[5-(oxan-4-ylmethyl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}ethan-1-one
N-[2-(piperazin-1-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-({1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
1-[benzyl(methyl)amino]-3-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-(1-ethyl-1H-1,2,4-triazol-5-yl)-3-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}benzamide
N2,N2-diethyl-N4-methyl-N4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]pyrimidine-2,4,6-triamine
1-{2-oxo-2-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethyl}-4-phenylpyrrolidin-2-one
4-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-2-(pyridin-4-yl)quinoline
4-methoxy-6-[2-(morpholin-4-ylmethyl)phenyl]quinazoline
4-(dimethyl-1,3-oxazole-4-carbonyl)-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
3-benzyl-N-[2-(2-fluorophenyl)ethyl]-1,2-oxazole-5-carboxamide
4-[4-(2-methylphenoxy)piperidin-1-yl]-6-(piperidin-3-yl)pyrimidine
(3aS,6aR)-5-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[3-({[2-(4-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}amino)propyl]pyrrolidin-2-one
N-methyl-N-(1-methylpyrrolidin-3-yl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
2-(benzyloxy)-N-(5-oxo-1-phenylpyrrolidin-3-yl)acetamide
N-[(3,4-dimethoxyphenyl)methyl]-3-ethyl-N-(1-methoxypropan-2-yl)-1,2-oxazole-5-carboxamide
N4-[(3S,4R)-4-methoxyoxolan-3-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
methyl 5-oxo-5-(3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}piperidin-1-yl)pentanoate
3-(4-methyl-1H-pyrazol-1-yl)-1-[4-(piperidine-1-carbonyl)piperidin-1-yl]propan-1-one
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-methyl-N-(1-methylpiperidin-4-yl)pyrimidine-5-carboxamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-{[3-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(4-{5-ethyl-6-methylthieno[2,3-d]pyrimidin-4-yl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(4-fluorophenyl)acetamide
[2-(methylsulfanyl)ethyl]({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
3-{5-[2-(4,5-dimethyl-1H-pyrazol-3-yl)ethyl]-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(prop-2-en-1-yl)-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
N-butyl-N,5-dimethyl-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-[(4-ethoxyphenyl)methyl]-4-(1H-pyrazol-1-ylmethyl)piperidine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-oxo-N-(propan-2-yl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}ethan-1-one
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(4-methylphenyl)ethan-1-one
1-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetyl]-4-phenoxypiperidine-4-carboxylic acid
N-tert-butyl-3-(3,4-dimethylbenzamido)-2-methylbenzamide
5-{4-[(3-ethyl-3-hydroxypiperidin-1-yl)methyl]phenoxymethyl}furan-2-carboxylic acid
1-cyclopentyl-5-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
2-methyl-N-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4,5,6,7-tetrahydro-1,3-benzothiazol-4-amine
N-[3-(2-methoxybenzamido)phenyl]-4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
1-({[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]amino}methyl)cyclohexan-1-ol
4-[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1-phenylpiperazin-2-one
4-(6-methoxy-2H-1,3-benzodioxol-5-yl)-3-methyl-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one