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5-[butyl(methyl)amino]-1-[(4-methoxyphenyl)methyl]azepan-2-one
(2E)-N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-3-(4-methoxyphenyl)prop-2-enamide
[(2S)-1-{5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}pyrrolidin-2-yl]methanol
6-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-2,3-dimethylquinoxaline
N-(pyridin-2-ylmethyl)-4-[6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(1-ethoxy-2-methylpropan-2-yl)-4-propylpyrimidine-5-carboxamide
ethyl(oxan-4-ylmethyl)[(1-propyl-1H-imidazol-2-yl)methyl]amine
methyl 3-(2-chlorobenzamido)-6-[(2-methylpiperidin-1-yl)methyl]thieno[2,3-b]pyridine-2-carboxylate
(2S,4S)-1-cyclopentyl-4-[2-(2,3-difluorophenyl)acetamido]-N-ethylpyrrolidine-2-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(4-fluorophenyl)-N-methylpropanamide
butyl(ethyl){[4-phenyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
4-{2-[5-(4-methoxy-2-methylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridine
2-fluoro-N-(1-{2-oxo-2-[4-(thiophene-2-carbonyl)piperazin-1-yl]ethyl}-1H-pyrazol-4-yl)benzamide
3-(2H-1,3-benzodioxole-5-carbonyl)-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
2-(4-methyl-1,3-oxazole-5-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
1-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}-2-(morpholin-2-yl)ethan-1-one
5-[(4-hydroxyphenyl)methyl]-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
3-[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-1-ethyl-3-methylpiperidine
2-(4-fluorophenyl)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine
2-(2,2-dimethylpropanamido)-N,5-dimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]thiophene-3-carboxamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-4-carboxamide
4-[4-(azetidine-1-carbonyl)phenyl]-2-methylbutan-2-ol
2-amino-4-(1,5-dimethyl-1H-pyrazol-4-yl)-6-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]pyridine-3-carbonitrile
7-(1-phenylcyclopropaneamido)-N-(prop-2-en-1-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
4,6-dimethyl-2-oxo-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,3,4-tetrahydropyrimidine-5-carboxamide
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-2-[3-(methoxymethyl)pyrrolidin-1-yl]pyridine
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-methoxypropan-1-one
1-{4-[(dimethylsulfamoyl)amino]phenyl}-N-[3-(pyridin-3-yl)propyl]piperidin-4-amine
2-(4-fluoro-3-methylphenyl)-2-{methyl[2-(1H-pyrazol-1-yl)ethyl]amino}acetic acid
(1R,5R)-3-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-(2-hydroxyethyl)-N-methyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
(2S,4S)-4-(2-cyanobenzamido)-N-ethyl-1-[3-(methylsulfanyl)propyl]pyrrolidine-2-carboxamide
N-(3-methoxyphenyl)-3-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-4-yl}propanamide
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]propanamide
2-(ethoxymethyl)-1-[5-(methoxymethyl)thiophene-2-carbonyl]pyrrolidine
1-cyclopentyl-4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperazin-2-one
2-{1-[(3-methoxyphenyl)methyl]-4-(quinolin-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-benzyl-N-(1,3-thiazol-2-ylmethyl)-5-(thiophene-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-butyl-8-[5-(methoxymethyl)furan-2-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-methyl-N-[2-(oxan-4-yl)ethyl]-1,2-oxazole-3-carboxamide
3-(pyridin-4-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
3-{[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-2-methyl-1,2,3,4-tetrahydroisoquinoline
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-amine
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-methyl-2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]acetamide
(1R,5R)-6-(cyclobutylmethyl)-N-phenyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-(4-methylpiperazin-1-yl)-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}pentan-1-one