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N-[2-(3-fluorophenyl)ethyl]-2-(4-{4-[methyl(oxan-4-yl)amino]piperidin-1-yl}phenyl)acetamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(propan-2-yl)piperidin-3-ol
N-(1-{7-[(5-ethylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-3,5-dimethylbenzamide
8-(3-fluoropyridin-2-yl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-cycloheptyl-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-methylurea
1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-amine
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-2-ylmethyl)amine
N-ethyl-2-[4-(propan-2-yl)piperazin-1-yl]pyrimidin-4-amine
(5-{1-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
1-{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
N-[(1-phenylcyclopentyl)methyl]-6-(pyrazine-2-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-methylurea
1-({4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-N,N-diethylpiperidine-3-carboxamide
2-[2-methyl-4-(2-propyl-1H-imidazol-1-yl)phenoxy]acetamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-4-oxo-4-phenylbutanamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(pyridine-4-carbonyl)piperidine-2-carboxamide
4-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)-N-(pyridin-3-yl)benzamide
5-(2,6-difluorophenoxymethyl)-N-(2,3-dihydro-1H-inden-2-yl)-1,2-oxazole-3-carboxamide
1-(4-phenylpiperazin-1-yl)-3-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}propan-1-one
2-cyclopropyl-9-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
(benzylsulfamoyl)[2-(1-methylpyrrolidin-2-yl)ethyl]amine
{[5-methyl-1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
7-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-(2-hydroxyethyl)-1-methyl-3-(trifluoromethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
N-[2-(1H-pyrazol-1-yl)ethyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
1-[1-({1-[3-(dimethylamino)benzoyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
6-(2-chlorophenyl)-2-(3-hydroxyazetidine-1-carbonyl)-7-(3-methylbut-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
[7-chloro-5-(1-methyl-1H-imidazol-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
(1S,4S)-2-(3-chlorophenyl)-5-[(2R)-oxolane-2-carbonyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
(2S,4R)-4-(3-chlorothiophene-2-amido)-N-methyl-1-[3-(methylsulfanyl)propyl]pyrrolidine-2-carboxamide
(4aS,8aR)-6-(dimethyl-1,3-oxazole-5-carbonyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(3-fluorophenyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1,3-benzoxazole-5-carboxamide
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-2-(1H-pyrazol-1-yl)acetamide
3-[2-({3-azaspiro[5.5]undecan-9-yl}amino)ethyl]-1,3-oxazolidin-2-one
N-({2-[(dimethylamino)methyl]phenyl}methyl)-4-hydroxy-N-methyl-2-(3-methylphenyl)pyrimidine-5-carboxamide
N-cyclobutyl-3-[(2-methyl-5-oxo-1,4-diazepan-1-yl)sulfonyl]benzamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(5-propyl-1,2-oxazole-3-carbonyl)-1,4-diazepane
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-[(5-methylfuran-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-methyl-1-(2-methylpropyl)-4-(1H-pyrrole-2-carbonyl)piperazin-2-one
5-{[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]methyl}pyrimidin-2-amine
N3-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
(3S,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
ethyl 3-[(3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidine-1-carbonyl)amino]propanoate
1-(2-methylquinolin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N,1,3-trimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(3S,4R)-1-(1-benzofuran-5-carbonyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
1-[4-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
5-methyl-2-[3-(morpholine-4-carbonyl)piperidin-1-yl]pyrimidin-4-amine