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1-methyl-3-[4-(4-{[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]imidazolidin-2-one
4-methyl-N-{3-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}benzene-1-sulfonamide
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N,N-diethyl-1H-pyrazole-4-carboxamide
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-(piperidin-1-ylmethyl)benzamide
1-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}cycloheptane-1-carboxamide
(butan-2-yl)({[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl})(thiophen-3-ylmethyl)amine
methyl N-[1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-1-oxopropan-2-yl]carbamate
7-chloro-4-[4-(piperidin-3-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-(4-methanesulfonylphenyl)quinoline
N-[4-(3-fluorophenyl)phenyl]-1-[(trimethylpyrazin-2-yl)methyl]piperidine-3-carboxamide
N3-tert-butyl-N5-[2-(4-methoxyphenyl)ethyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
7-(2,3-dihydro-1-benzofuran-5-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-methyl-3-(pyrrolidin-1-yl)propyl]amine
2-[(3-{[(2,3-dimethylphenyl)methyl]carbamoyl}phenyl)amino]acetic acid
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
1'-(4,6-dimethylpyridine-3-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
1-(2-chlorophenyl)-4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperazin-2-one
8-(3-ethyl-1H-pyrazole-4-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[2-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-2-oxoethyl]-1,2,3-oxadiazol-3-ium-5-olate
N-cyclopropyl-1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
5-chloro-2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
2-(4-methyl-1,4-diazepan-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
N-[4-(3-methylpyrazin-2-yl)phenyl]methanesulfonamide
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-[(2-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)acetamide
4-(5-methylpyridin-2-yl)-1-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]piperidin-4-ol
N-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
N-(propan-2-yl)-4-{[4-(pyridin-4-yl)piperazin-1-yl]sulfonyl}benzamide
N-(1,2-oxazol-3-ylmethyl)-7-(1,3-thiazole-5-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(3-benzamido-4-methoxyphenyl)-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
(2S,4S)-N-ethyl-1-[(3-methylthiophen-2-yl)methyl]-4-(thiophene-3-amido)pyrrolidine-2-carboxamide
5-[3-(methoxymethyl)piperidine-1-carbonyl]-2-[4-(1H-pyrazol-5-yl)phenyl]pyridine
4-{[3-(piperidine-1-carbonyl)-1-[3-(pyridin-3-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoline
1-(3-chloro-4-methylbenzoyl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine
1-(4,4-difluoropiperidin-1-yl)-2-(dimethylamino)-2-(2-methylphenyl)ethan-1-one
3-[1-tert-butyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]pyridine
4-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-6-methylpyrimidin-2-amine
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(naphthalene-1-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{1-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-amine
8-(3-ethyl-1H-pyrazole-5-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(6-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl)morpholine
2-tert-butyl-6-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-(azepane-1-sulfonyl)-5-[2-(hydroxymethyl)phenyl]benzoic acid
3-{2-[5-(1-ethyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,3-oxazolidin-2-one
6-[(2-fluorophenyl)methoxy]-4-(5-methyl-1H-pyrazole-3-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
4-amino-5-(2,1,3-benzothiadiazol-4-yl)-2-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[2,3-d]pyrimidin-7-one
N-(3-chloro-4-fluorophenyl)-3-[1-(3-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]propanamide