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1-[9-benzyl-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-methoxyethan-1-one
1-cyclopentyl-5-oxo-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]pyrrolidine-3-carboxamide
3-(3-methoxyphenyl)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1H-pyrazole-5-carboxamide
4-ethyl-3-{[1-(5-methyl-1H-1,3-benzodiazole-2-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,3R)-2-{[5-(2,4-difluorophenoxymethyl)-1,2-oxazol-3-yl]formamido}-3-hydroxybutanamide
1-cyclopentyl-4-(2-methyl-1,8-naphthyridine-3-carbonyl)piperazin-2-one
2-[2-(2-methoxyquinolin-3-yl)-4-methylphenoxy]acetamide
[(1-cyclopentylpiperidin-4-yl)methyl][(8-methoxy-2H-chromen-3-yl)methyl](pyridin-3-ylmethyl)amine
1-{4-[3-(difluoromethoxy)benzoyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
2-{[3-(morpholin-4-yl)propyl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyrimidin-4-amine
3-methyl-5-{1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidin-2-yl}-1,2-oxazole
1,7-dimethyl-2-[2-(piperidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-indole
N-benzyl-4-(1-methyl-6-oxo-1,6-dihydropyridazin-3-yl)benzene-1-sulfonamide
1'-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)acetamide
2-[2-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
3-[5-(5-methylpyrazine-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-(4-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-oxobutan-2-yl)acetamide
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-2-methylphenyl)urea
4-(5-fluoro-3-methyl-1H-indole-2-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
8-(2-methoxyethyl)-N-(2-methoxyphenyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
ethyl 1-(3-methylbutyl)-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(3-{1-[2-(morpholin-4-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyridine-3-carbonitrile
11-(benzylamino)-4-cyclopentyl-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(5-acetylthiophen-3-yl)-1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]ethan-1-one
1-[1-(cyclopropylmethyl)-7-oxoazepan-4-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
7-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
4-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}thiomorpholine
N-{1-[4-(4-methoxyphenoxy)piperidin-1-yl]-1-oxopropan-2-yl}methanesulfonamide
5-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-3-yl}-N-[(2-methoxyphenyl)methyl]-4-methyl-1,3-thiazol-2-amine
5-[1-cyclohexyl-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]-1-methyl-1,2-dihydropyridin-2-one
2-(3-hydroxypropyl)-8-{[4-(methylsulfanyl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
6,7-dimethoxy-2-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}quinazolin-4-amine
ethyl 4-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-3-yl]piperazine-1-carboxylate
4-benzyl-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}pyrrolidin-2-one
3-[(3R,4S)-1-(1,3-benzothiazol-2-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1-(2-amino-5-ethylpyrimidin-4-yl)-3-ethylpiperidin-3-ol
1-ethyl-3-methyl-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]piperidine-3-carboxamide
5-{[(3S)-3-(dimethylamino)pyrrolidin-1-yl]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-ethyl-N-(oxan-4-yl)-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-({3-methyl-7-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-5-carboxamide
(2R,6R)-4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-[(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)amino]pyridine-3-carboxamide
N-({1-[(3-methylphenyl)methyl]-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl}methyl)acetamide
ethyl 1-(2-phenoxyacetyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
[(2,4-dimethoxyphenyl)methyl](methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-methyl-6-{[3-(morpholine-4-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2,3,4-tetrahydroquinoline
5-[2-(ethylamino)ethyl]-1-[3-(propan-2-yloxy)propyl]pyrrolidin-2-one
2-[4-(dimethylamino)azepan-1-yl]-4,6-dimethylpyridine-3-carbonitrile