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2-(2-amino-2-methylpropanoyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-[(3S,4R)-1-(5-fluoropyridin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
ethyl 4-[(4-{[1-(furan-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
N-{[2-(3-hydroxypiperidin-1-yl)-7-methylquinolin-3-yl]methyl}-2-methoxy-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
1-(3-methanesulfonamido-4-methoxyphenyl)-3-[1-(thiophen-2-yl)propan-2-yl]urea
1-[2-(4-fluoro-2-methylphenyl)acetyl]-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
3-[5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)pyridin-2-yl]benzoic acid
N-(5-chloro-2-methoxyphenyl)-3-(morpholin-4-yl)piperidine-1-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(4-fluorobenzenesulfonyl)ethyl]acetamide
[(3R,4R)-1-(2,3-dihydro-1H-indene-5-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-tert-butyl-3-{[(2-fluorophenyl)methyl]amino}-5-(4-methyl-1,4-diazepane-1-carbonyl)benzene-1-sulfonamide
5-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
N-(2,3-dihydro-1H-inden-2-yl)-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-4-methylpyridine-3-carboxamide
7-(3-chlorophenyl)-4-[3-(1H-pyrazol-1-yl)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(3-hydroxypropyl)-9-(1H-indole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
5-(cyclopropylmethyl)-2-(3,4-difluorophenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
5-ethyl-N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-[3-(4-fluorophenyl)phenyl]-1-propanoylpiperidine-3-carboxamide
[3-(2-phenylethyl)-1-[3-(trifluoromethyl)benzoyl]piperidin-3-yl]methanol
2-{1-[(2-methylphenyl)methyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
3-(4-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrazine-2-carbonitrile
1-(4-methyl-3-phenylpiperazin-1-yl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
N,N-dimethyl-6-{4-[(thiophen-2-ylmethoxy)methyl]phenyl}pyridazin-3-amine
3-methyl-N-[4-(5-methylfuran-3-amido)phenyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(3-hydroxypropyl)-2,4-dimethyl-N-[(5-methylthiophen-2-yl)methyl]-1,3-thiazole-5-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(3-fluoropyridin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-ethoxy-3-{[4-(4-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
{3-methyl-1-[4-(3-methylphenoxy)piperidin-1-yl]-1-oxobutan-2-yl}urea
{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)propylamine
2-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline
3-chloro-N-cyclopentyl-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
5-(azocane-1-carbonyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
1-[2-(4-methoxyphenyl)ethyl]-8-(2-methylpropyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-hydroxy-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
ethyl 4-(2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperazine-1-carboxylate
6-cyclopentyl-1-methyl-N-[(3-propyl-1,2-oxazol-5-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-cyclobutylacetamide
1-(cyclohexylmethyl)-4-[(thian-4-yl)amino]pyrrolidin-2-one
(1S,5R)-6-(morpholine-4-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-[3-(dimethylsulfamoyl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2,1-benzoxazole-3-carboxamide
3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}-N-(thiophen-2-ylmethyl)aniline
N-[3-(furan-2-yl)phenyl]-1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}piperidine-4-carboxamide
1-[(4-benzyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]-N,N-diethylpiperidine-3-carboxamide
1-[3-(pyridin-3-yl)azetidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
7-[(3-methylphenyl)methyl]-2-(propane-2-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
[5-({4-[(4-methylphenyl)sulfanyl]piperidin-1-yl}methyl)furan-2-yl]methanol