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5-[3-(3-methyl-1H-1,2,4-triazol-5-yl)propanoyl]-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
8-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{1'-[(5-acetylthiophen-3-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
1'-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]
2-methyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,3-benzothiazole-6-sulfonamide
3-(1-butyl-1H-imidazol-2-yl)-N-(2-fluorophenyl)piperidine-1-carboxamide
N-(1-{1-[3-(furan-2-yl)propanoyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-6-methoxy-N,3-dimethyl-1-benzofuran-2-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide
1-(3-chlorophenyl)-4-[2-(methylsulfanyl)pyridine-3-carbonyl]piperazin-2-one
N-[1-(furan-2-yl)ethyl]-N-methyl-3-propyl-1H-pyrazole-5-carboxamide
(2S,4S)-4-(3,3-dimethylbutanamido)-N-ethyl-1-(3-methylthiophene-2-carbonyl)pyrrolidine-2-carboxamide
9-[(2,3-dichloro-4-methylphenyl)methyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
2-(1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}pyrrolidin-2-yl)-4-methyl-1H-1,3-benzodiazole
2-ethyl-4-methyl-N-[2-(4-sulfamoylphenyl)ethyl]-1,3-oxazole-5-carboxamide
(1R,5S,8S)-3-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-8-methoxy-3-azabicyclo[3.2.1]octane
1-{2-oxo-2-[3-(pyridin-4-yl)azetidin-1-yl]ethyl}imidazolidine-2,4-dione
1-[(3-methoxyphenyl)methyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-cyclopropyl-N-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1,3-benzothiazole
6-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-2-methyl-2,3-dihydropyridazin-3-one
3-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}-1,3-oxazinan-2-one
(3R,5S)-5-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}pyrrolidin-3-ol
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrrolidin-3-yl]methanol
2-{7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}propane-1,3-diol
(1R,5R)-6-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-ethoxy-5-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}pyridine
N-[3-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
3-{[(2S,5R)-5-{[(furan-3-ylmethyl)(methyl)amino]methyl}oxolan-2-yl]methyl}-N,N-dimethylbenzamide
1-[(4-fluorophenyl)methyl]-4-[2-(thiomorpholine-4-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
5-(4-chloro-3-fluorophenyl)pyrazin-2-amine
3-chloro-5-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]-1,2-dihydropyridin-2-one
(1R,9S)-5-amino-3-(7-methoxy-2H-1,3-benzodioxol-5-yl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-[2-(oxolan-3-yl)ethyl]-1,2-dihydroquinoxalin-2-one
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]propanamide
N-{1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-2-[2-(methoxymethyl)pyrimidin-5-yl]quinoline
2-(4-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)pyridine-3-carbonitrile
N-(1-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-5-(methoxymethyl)furan-2-carboxamide
4-[(benzyloxy)methyl]-1-[(5-methyl-1H-pyrazol-3-yl)methyl]-1H-1,2,3-triazole
1-cyclopropyl-6-oxo-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine-3-carboxamide
1-{imidazo[1,2-b]pyridazin-6-yl}-4-(3-phenylpropyl)piperazine
N-{3-[2-(2-methoxyphenyl)-1H-imidazol-1-yl]propyl}pyridin-3-amine
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(3-methylthiophene-2-carbonyl)pyrrolidin-3-yl]methanol
3-methyl-1-{1-[6-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
4-(2-methyl-2-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}propyl)morpholine
(4aR,7aS)-1-(cyclopropylmethyl)-4-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3aR,6aR)-2-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(2-methoxyethyl)-5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazole