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N-methyl-2-(4-propanoylphenoxy)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-ethyl-4-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
(2S,4S)-1-benzyl-4-{[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-(3-hydroxypropyl)-9-[(1-methyl-1H-indol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
4,6-dimethyl-2-oxo-N-{[5-(pyridin-2-yl)thiophen-2-yl]methyl}-1,2,3,4-tetrahydropyrimidine-5-carboxamide
{4-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
2-(ethylamino)-4-methyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,3-thiazole-5-carboxamide
1-{2-[(2,6-dichlorophenyl)methyl]-4-hydroxypyrimidine-5-carbonyl}piperidine-3-carboxylic acid
2-[3-methyl-4-({4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}methyl)-1H-pyrazol-1-yl]ethan-1-ol
N-[(3S,4R)-4-(4-methylphenyl)-1-(pyridine-3-sulfonyl)pyrrolidin-3-yl]acetamide
11-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
2-(azocan-1-yl)-1-[(3S)-3-ethylmorpholin-4-yl]ethan-1-one
(1R,3S)-3-methoxy-7-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-7-azaspiro[3.5]nonan-1-ol
6-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-indole
4-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
1-{2-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}piperidin-2-one
7,7-dimethyl-2-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(benzylsulfamoyl)[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]methylamine
4-[7-(1H-imidazole-2-carbonyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
methyl 4-[4-(3-fluoropyridin-4-yl)piperazin-1-yl]benzoate
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
8-(2,4-difluoro-3-methoxybenzoyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-amino-1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]ethan-1-one
4-({4-methyl-5-[1-(6-methylpyridine-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
4-{[1-cyclohexyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiane-1,1-dione
N-(1-carbamoylcyclopentyl)-2,6-dimethylpyridine-4-carboxamide
1-[3,5-dimethyl-1-(3-propanoylphenyl)-1H-pyrazol-4-yl]propan-2-one
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-(3,3-dimethylcyclohexyl)piperidine
2-amino-3-ethyl-N-methyl-N-(thian-4-yl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(ethoxymethyl)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[4-(2-aminopyrimidin-4-yl)-1H-pyrazol-1-yl]-N-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-5-yl}acetamide
N-[3-(2-oxopyrrolidin-1-yl)propyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
N-methyl-N-(pyridin-2-ylmethyl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,5-dimethylpyrazine-2-carboxamide
1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,2,3,4-tetrahydroquinolin-2-one
2-(furan-2-yl)-5-{1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-imidazol-2-yl}pyrimidine
1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-3-(thiophen-2-yl)propan-1-one
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-ethyl-N-(2-hydroxyethyl)-5-methyl-1H-pyrazole-4-carboxamide
2-methoxy-1-{4-methyl-2-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]piperazin-1-yl}ethan-1-one
3-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridin-2-amine
1-(azepan-1-yl)-3-[3-({[3-(pyridin-3-yloxy)propyl]amino}methyl)phenoxy]propan-2-ol
(2S,4R)-4-amino-1-[(8-methoxyquinolin-2-yl)methyl]-N-methylpyrrolidine-2-carboxamide
5-methyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]pyrazine-2-carboxamide
1-(azepan-1-yl)-3-[3-({[3-(dimethylamino)propyl](methyl)amino}methyl)phenoxy]propan-2-ol
(1R,5R)-3-(1-benzyl-1H-pyrazole-4-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methylacetamide