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8-(3,4-dimethylbenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[2-(4-methoxyphenyl)ethyl]-2-methyl-N-[(1-methylpiperidin-4-yl)methyl]-1H-pyrrole-3-carboxamide
(2R,6S)-4-{1-[(2,3-difluoro-6-methoxyphenyl)methyl]piperidin-4-yl}-2,6-dimethylmorpholine
1-(4-aminopyrimidin-2-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylic acid
6-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1H-pyrazole-4-carboxamide
2-[4-(hydroxymethyl)phenyl]-1-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
2-[(3R,5R)-5-(morpholine-4-carbonyl)piperidine-3-carbonyl]-2,3-dihydro-1H-isoindole
3-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(3-phenylphenyl)-N-[2-(pyridin-3-yl)ethyl]piperidin-4-amine
2-(5-methyl-1H-pyrazole-3-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
5-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1-[(2-methoxyphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
2,4-difluoro-6-(2-methoxyquinolin-3-yl)phenol
(4aS,7aR)-1-acetyl-4-benzyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aR,7aS)-1-cyclobutanecarbonyl-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-3-methyl-6-(naphthalene-1-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(furan-3-ylmethyl)-N-methyl-4-(piperidin-3-ylmethyl)benzamide
1-ethyl-4-{2-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}piperazine-2,3-dione
4-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}thiomorpholine
1-[(4-chlorophenyl)methyl]-6-oxopiperidine-3-carboxylic acid
6-amino-2-(2-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}ethyl)pyrimidin-4-ol
N-[2-(5-methylfuran-2-yl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
ethyl 4-({[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}amino)piperidine-1-carboxylate
2-(4-chloro-2-{[4-(oxan-4-yl)piperazin-1-yl]methyl}phenoxy)acetic acid
N-[1-({1-[(3,5-dimethylphenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)-1H-pyrazol-5-yl]acetamide
N,1-dimethyl-N-[(3-methyloxetan-3-yl)methyl]-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(1,2-benzoxazol-6-yl)-1-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}urea
6-ethyl-N-[2-(7-methyl-1H-indol-3-yl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
1-({1-[3-(2-methoxyphenyl)benzoyl]pyrrolidin-2-yl}methyl)-1H-pyrazole
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-(4-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenyl)-3,4,5,6,7,8-hexahydroquinazolin-4-one
(1R,5S,6R)-3-cyclopentyl-N-[2-(1H-imidazol-1-yl)ethyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
1-[2-methoxy-6-({[(1-methylpiperidin-4-yl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)acetamide
2-(2-chlorophenyl)-N-(2-hydroxyethyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2,5-dimethylpyrazine
3-{[(4-chlorophenyl)methyl]({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl})amino}propan-1-ol
3-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(propan-2-yl)propanamide
6-amino-2-{2-[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]ethyl}pyrimidin-4-ol
1-(2,3-dihydro-1H-inden-2-yl)-4-(2-ethylpyridine-4-carbonyl)-1,4-diazepane
2-tert-butyl-N-[4-(1H-pyrazol-1-yl)phenyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
1-(5-{[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
(2E)-N-({3-methyl-7-[2-(pyrrolidin-1-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenylprop-2-enamide
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-cyclohexyl-1,4-diazepane
{3-[(4-fluorophenyl)methyl]-1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-yl}methanol
1-[(4-{[5-(methoxymethyl)furan-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
methyl[2-(2-methylpiperidin-1-yl)ethyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
methyl 6-{[butyl(methyl)amino]methyl}-3-(2-chlorobenzamido)thieno[2,3-b]pyridine-2-carboxylate
3-{[(1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine