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1-{4-[2-(3-methoxyphenyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
1-[2-(dimethylamino)-6-(1H-imidazol-2-ylmethyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
2-methoxy-3-(5-methoxypyridin-3-yl)pyridine
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(1H-pyrrole-2-carbonyl)piperazine
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)butanamide
2-(2-hydroxyethyl)-9-{[3-(trifluoromethyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
(3R,4R)-4-ethyl-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidine-3,4-diol
(3S,9aR)-3-(1H-indol-3-ylmethyl)-8-(2-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1S,5R)-3-[(dimethylcarbamoyl)methyl]-N-[(4-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-[2-(2-hydroxyethoxy)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperazine
N-(pyridin-4-ylmethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
2-(5-acetylthiophen-3-yl)-N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]acetamide
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]ethan-1-one
{[5-(2-chlorophenyl)furan-2-yl]methyl}(methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
1-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
4-[(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-3-yl)methyl]benzoic acid
3-(3,4-dimethoxybenzoyl)-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine
(1R,5S,6S)-6-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
3-(2H-1,3-benzodioxol-5-yl)-5-[(5-methylthiophen-2-yl)methyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-(5-chloro-2-methylphenyl)-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazine
N,N-diethyl-2-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]acetamide
2-(dimethylamino)-1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(2-methylphenyl)ethan-1-one
3-(4-chloro-1H-pyrazol-1-yl)-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]propan-1-one
(2S)-2-[(4-methylpiperidin-4-yl)formamido]-3-phenylpropanamide
N-cyclopropyl-1-(1-{[(1-methyl-1H-pyrazol-3-yl)carbamoyl]methyl}piperidin-4-yl)piperidine-3-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
1-(3-{4-[2-(3-methylphenyl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}propyl)pyrrolidin-2-one
5-(2,3-dihydro-1-benzofuran-2-carbonyl)-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-{2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
ethyl 4-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine-1-carboxylate
N5,N5,N6-trimethyl-N6-[(3-methyl-1H-indol-2-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1-(6-methoxyquinolin-8-yl)urea
3-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]carbamoyl}amino)-4-methoxy-N-methylbenzamide
5-tert-butyl-4-[(2,6-dioxo-1,3-diazinan-1-yl)methyl]furan-2-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
methyl 4-{[2-(5-acetylthiophen-3-yl)acetamido]methyl}benzoate
1-cyclohexyl-4-(6-methoxypyridin-3-yl)-3-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-(4-chlorophenyl)-1-{[2-hydroxy-5-(pyrimidin-2-yl)phenyl]methyl}piperidin-4-ol
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(pyridin-4-yl)ethan-1-one
4-(3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propoxy)benzamide
(3R,5S)-N3-(4-fluorophenyl)-1-(pyridin-4-ylmethyl)-N5-(thiophen-2-ylmethyl)piperidine-3,5-dicarboxamide
7,7-dimethyl-2-(pyrimidin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
methyl[(6-methylpyridin-2-yl)methyl][(3-phenyl-1,2-oxazol-5-yl)methyl]amine
N-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
N-[3-(4-methylpiperazine-1-carbonyl)phenyl]azocane-1-carboxamide
N-{[3-(difluoromethoxy)phenyl]methyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[(3R,5S)-1-(cyclopentylmethyl)-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-{[5-oxo-1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,2-oxazole-3-carboxamide