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4-benzyl-3-{1-[2-(propan-2-yloxy)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyloxan-4-amine
2-(1-benzyl-4-cyclopentylpiperazin-2-yl)ethan-1-ol
4-fluoro-N-({1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}methyl)benzamide
6-methyl-5-{5-[2-methyl-5-(propan-2-yl)furan-3-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-[(3R,4S)-1-[(methylcarbamoyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-1,2,3,4-tetrahydroquinoline-8-carboxamide
2-(4-{[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenoxy)ethan-1-ol
N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
2-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
6,7-dimethyl-4-({[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-2H-chromen-2-one
1-(cyclopropylmethyl)-5-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-ethyl-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
4-{3-[(4aR,8aR)-octahydro-2H-1,4-benzoxazine-4-carbonyl]phenyl}-2-methylbutan-2-ol
N,N-dimethyl-5-[(2-phenylethyl)amino]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3ar,6ar)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-(pyridin-2-yl)pyrimidin-2-amine
2-amino-6-[4-(morpholin-4-yl)phenyl]-4-(pyridin-3-yl)pyridine-3-carbonitrile
6-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(1H-indol-3-yl)-N-methylacetamide
(3aS,6aR)-3-cyclopentyl-5-[(trimethylpyrazin-2-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-hydroxy-2-(4-methoxyphenyl)ethan-1-one
(4aR,7aS)-1-methyl-4-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N3-tert-butyl-4-oxo-N5-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(3S)-1,3-dimethyl-4-{6-[(thiophen-2-ylmethyl)amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}piperazin-2-one
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
3-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-3-yl)-N-[4-(trifluoromethyl)phenyl]propanamide
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1-methylimidazolidin-2-one
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(2R,3R)-2-ethoxy-1'-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-[3-(dimethylamino)propyl]-N-methyl-1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-amine
2-[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amino]-N-(pyrazin-2-yl)acetamide
(2S,4R)-4-amino-N,N-diethyl-1-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyrrolidine-2-carboxamide
4-(2-methyl-1,6-naphthyridine-3-carbonyl)piperazin-2-one
diethyl({[3-(3-phenylpiperazine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(3-fluoropyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(3,5-dimethylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N,N-dimethyl-4-{[5-(oxan-2-yl)furan-2-yl]methyl}piperazine-1-sulfonamide
N-cycloheptyl-2-[(3R,4S)-3-methanesulfonamido-4-(propan-2-yl)pyrrolidin-1-yl]acetamide
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-[3-(2-methyl-1H-imidazol-1-yl)propyl]piperazin-2-one
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)piperidin-2-one
N,N-dimethyl-2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-4-amine
N-(2-{3-methyl-7-oxo-7H-[1,3]thiazolo[3,2-b][1,2,4]triazin-6-yl}phenyl)-1H-1,2,4-triazole-5-carboxamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
(3S,4S)-4-cyclopropyl-1-[4-(4-fluorophenyl)butanoyl]pyrrolidine-3-carboxylic acid
5-(4-methoxyphenyl)-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]-1,2,4-triazin-3-amine