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4-methyl-5-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
1-(diphenylmethyl)-4-(4-methyl-1,3-oxazole-5-carbonyl)piperazine
3-chloro-5-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
ethyl 1-[5-methyl-2-(propylamino)benzoyl]piperidine-3-carboxylate
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methoxyphenoxy)acetamide
2-[3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
5-{1-[2-(4-methoxyphenyl)ethyl]-1H-pyrazol-3-yl}-4-methyl-N-(thiophen-3-ylmethyl)-1,3-thiazol-2-amine
N-[3-(1H-imidazol-1-yl)butyl]-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[3-(pyridine-2-carbonyl)piperidin-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
1-(4-{5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-diazepan-1-yl)ethan-1-one
N-cyclopentyl-5-(2,2-dimethylpropyl)-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(2,3-dihydro-1H-isoindole-2-carbonyl)-2-[2-(2-methoxyethyl)pyrimidin-5-yl]quinoline
3-{5-[3-(2-methylphenyl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
5-methyl-5-(4-methylpent-3-en-1-yl)-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]piperidin-2-one
{3-[5-(2,3-difluoro-4-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]propyl}dimethylamine
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-2-(1H-pyrazol-1-yl)acetamide
4-{4-[(cyclopropylcarbamoyl)amino]phenyl}-N,N-dimethylbenzamide
2-[1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1H-imidazol-2-yl]pyridine
4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-2-(thiophen-3-yl)-1,3-oxazole
1-{6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}-1,4-diazepan-5-one
3-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-3-(3-fluorophenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
3-[3-(piperazin-1-ylmethyl)phenyl]benzoic acid
1-[6-(2-aminoethyl)pyrimidin-4-yl]-4-phenylpiperidine-4-carbonitrile
1-{1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}butan-1-one
3-(3-methoxypropyl)-1-(4-methoxypyrimidin-2-yl)piperidine-3-carboxylic acid
(1R,5R)-6-[(4-chloro-3-fluorophenyl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(5-amino-1,3,4-thiadiazol-2-yl)-1-[2-(3-phenylpropyl)morpholin-4-yl]ethan-1-one
2-(carbamoylamino)-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}acetamide
2-fluoro-5-[3-(1H-pyrazol-3-yl)phenyl]benzoic acid
2-cyclopentyl-9-[5-(methoxymethyl)furan-2-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
N-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}pyrimidin-4-amine
[(5-{[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}thiophen-3-yl)methyl]dimethylamine
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-methyl-1,2,3-thiadiazole-5-carboxamide
N-[(2S,4R,6S)-2-benzyl-6-[2-methyl-1-(morpholin-4-yl)propan-2-yl]oxan-4-yl]acetamide
2-{3-[6-(hydroxymethyl)-1,4-oxazepane-4-carbonyl]phenoxy}-1-(piperidin-1-yl)ethan-1-one
(1S,5R)-6-(cyclopropylmethyl)-N-(2,5-dimethylphenyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methanol
7-(3-chlorophenyl)-4-(1-methylcyclopropanecarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2-methoxyacetyl)-4-[(methylcarbamoyl)methyl]-1,4-diazepane-6-carboxylic acid
{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-pyrazol-4-yl)ethyl]amine
4-[(4-fluorophenyl)sulfanyl]-6-[2-(trifluoromethyl)morpholin-4-yl]pyrimidin-2-amine
2-(2,3-difluorophenoxymethyl)-N-methyl-N-[(4-methylphenyl)methyl]-1,3-oxazole-4-carboxamide
2-{[3-(cyclopropylcarbamoyl)piperazin-1-yl]methyl}-3,5-dimethoxybenzoic acid
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-methoxy-N-methylpyridine-3-carboxamide
2,2-diethyl-4-{5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}morpholine
(1R,9aR)-1-({[(2-ethoxy-3-methoxyphenyl)methyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
7-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}-N-propylpyrazolo[1,5-a]pyrimidine-6-carboxamide
methyl 2-({3-[4-(pyridin-3-yl)piperazine-1-carbonyl]phenyl}amino)acetate
7-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one