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2-(2-phenylethyl)-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]morpholine
3-(4-ethyl-1H-pyrazol-5-yl)-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidine
4-(benzyloxy)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzamide
7-(2-methoxyethyl)-2-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-2,7-diazaspiro[4.5]decane
4-{[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
1-{1-[4-(dimethylamino)benzoyl]piperidin-3-yl}-3-phenylpropan-1-one
1-(4-fluoro-3-methylbenzoyl)-3-(3-methylphenoxy)azetidine
6-ethyl-2-(morpholin-4-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyrimidin-4-amine
N-({1-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]piperidin-4-yl}methyl)acetamide
1-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(1H-pyrazol-1-yl)butan-1-one
1-[2-({[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}amino)ethyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one
5,8-dimethyl-2-[({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amino)methyl]quinolin-4-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(thiophene-2-carbonyl)piperidin-3-ol
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
N-(1-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylfuran-2-carboxamide
N-{[1-(4-chlorophenyl)cyclopropyl]methyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
ethyl({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}){[3-(methylsulfanyl)phenyl]methyl}amine
1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-2-(1H-1,2,4-triazol-3-ylsulfanyl)ethan-1-one
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-methoxyethyl)-1,3-dimethyl-1H-pyrazole-4-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(5-methylfuran-2-yl)methyl]-1,3-oxazole-4-carboxamide
(2S)-2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidine
N-(1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N,2-dimethylfuran-3-carboxamide
N-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-1-methyl-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
methyl 1-[(3R,5S)-1-(adamantan-2-yl)-5-[(thiophen-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine
2-amino-N-(2-oxoazepan-3-yl)-4-phenylpyrimidine-5-carboxamide
6-tert-butyl-N,1-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-methyl-9-(morpholine-4-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-({1-[(6-chloro-2-fluoro-3-methylphenyl)methyl]piperidin-3-yl}methyl)methanesulfonamide
{3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-5-methyl-1,2-oxazol-4-yl}methanol
(1S,9R)-11-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
(3S,4S)-1-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
[(3R,4R)-1-[(3-ethenylphenyl)methyl]-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
1-[2-(1H-pyrazol-1-yl)acetyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
1-methyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
methyl 2-{[2-(cyclohex-1-en-1-yl)ethyl]sulfamoyl}-6-(1-methyl-1H-pyrazole-3-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
N-[(2,4-difluorophenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-benzyl-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-1,3-thiazole-4-carboxamide
N-(3-cyanothiophen-2-yl)-3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}benzamide
(3aR,6aR)-2-(4-methoxy-2-methylbenzoyl)-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}-1-{[1-(pyridin-2-yl)piperidin-3-yl]methyl}urea
2-phenoxy-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
3-benzyl-4-(4-propylpyrimidine-5-carbonyl)piperazin-2-one
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-[1-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
1-methyl-2-oxo-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)-1,2-dihydropyridine-3-carboxamide