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methyl 1-({6-oxo-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)piperidine-2-carboxylate
1-{2-[({4-[3-(azepan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]ethyl}pyrrolidin-2-one
N-cyclopropyl-2-(4-propanoylphenoxy)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
2-{[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}benzonitrile
N-cyclobutyl-2-(2-methoxybutanoyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
6-(2,5-dimethoxybenzoyl)-7-methyl-4-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
3-(2-{3-[5-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1,3-benzoxazol-2-one
4-[2-(4-fluoro-3-methylphenyl)acetyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methylpentanamide
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-(4-phenylpiperidin-1-yl)acetamide
2-(1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carbonyl)pyridine
4-{2-[1-(quinoxaline-2-carbonyl)piperidin-2-yl]ethyl}phenol
6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
(2S,4R)-4-amino-N,N-diethyl-1-(1-methylcyclopropanecarbonyl)pyrrolidine-2-carboxamide
1-cyclopropyl-4-[5-(pyridin-3-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
cyclopentyl 4-[({[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}carbamoyl)amino]benzoate
2-[2-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)phenoxy]acetamide
1-methanesulfonyl-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
N-[(3S)-1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl]acetamide
(2S,4S)-1-(2,5-dimethylfuran-3-carbonyl)-N,N-diethyl-4-(3-hydroxypropanamido)pyrrolidine-2-carboxamide
5-[3-(dimethylamino)pyrrolidine-1-carbonyl]-N-ethylpyrimidin-2-amine
4-methyl-2-(2-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one
1-(1-{3-benzyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}propyl)-1H-pyrazole
(3S,4S)-4-methyl-1-(5-methylthiophene-2-carbonyl)piperidine-3,4-diol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N,N-diethyl-1-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
2-[4-(acetamidomethyl)-1,2,3,6-tetrahydropyridin-1-yl]-N-[1-(4-methylphenyl)ethyl]acetamide
4-{3-[2-(4-phenyl-1H-imidazol-5-yl)phenoxy]propyl}morpholine
2-(azepan-1-yl)-N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}acetamide
{[6-(2-ethoxyphenyl)pyridin-3-yl]methyl}dimethylamine
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}benzamide
3-{[(1-hydroxybutan-2-yl)(pyridin-2-ylmethyl)amino]methyl}phenol
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
3-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-1-(4-ethylpiperazin-1-yl)propan-1-one
3-(1H-imidazol-1-ylmethyl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine
1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-[4-(furan-2-yl)phenyl]piperidine-3-carboxamide
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
(2S,4S)-N-[2-(dimethylamino)ethyl]-1-[(3-fluorophenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carboxamide
(2S)-2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-3-methylbutanamide
5-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-(oxan-4-yl)piperidine-4-carboxamide
(1S,5R)-3-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-2-oxo-N-phenyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
1-[2-(2-methoxypyridin-3-yl)pyrimidin-4-yl]piperidin-4-ol
1-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}cyclopropane-1-carboxamide
1-(2-methoxyphenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
4-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2-methoxyphenyl)piperazin-2-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-(4-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
2-(3,5-dichloro-4-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
8-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one