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{[2-(azocan-1-yl)pyridin-3-yl]methyl}(thiophen-2-ylmethyl)amine
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]ethan-1-one
3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-diazinane-2,4-dione
[5-({methyl[1-(3-methylpyridin-2-yl)propan-2-yl]amino}methyl)furan-2-yl]methanol
N-({5-[(2,6-difluoro-3-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
2-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)-N-(propan-2-yl)acetamide
6-methyl-2-{1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
N,N-diethyl-3-(2-methylquinazolin-4-yl)benzamide
4-({1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)-1-methylpiperazin-2-one
N-methyl-2-{4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}propanamide
1-[(4-chlorophenyl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-1,2,5-thiadiazole-3-carboxamide
1-(2-aminoethyl)-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-methyl-4-phenylpiperazine
dimethyl[2-({[1-(propan-2-yl)piperidin-4-yl]methyl}(thiophen-3-ylmethyl)amino)ethyl]amine
N-tert-butyl-2-(2-ethyl-6-methylpyrimidin-4-yl)benzene-1-sulfonamide
2-{[2-(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)-1H-imidazol-1-yl]methyl}-3,4-dihydroquinazolin-4-one
2-(3-{3-[4-(1H-imidazol-1-ylmethyl)phenyl]phenyl}-1H-pyrazol-1-yl)ethan-1-ol
2-methoxy-1-{3-[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-one
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-phenylmethanesulfonylpyrrolidin-3-amine
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(methylsulfanyl)propan-1-one
3-(4-hydroxy-3-methoxyphenyl)-4-(3-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-acetyl-1,4-diazepan-1-yl)-2-[4-(benzyloxy)phenyl]acetic acid
(2E)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-4-methyl-N-(oxolan-2-ylmethyl)pent-2-enamide
3-{[(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)oxy]methyl}pyridine
2-(hydroxymethyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{5-[4-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
5-(4-cyclohexylphenyl)-N-[1-(pyrimidin-4-yl)ethyl]-1,2,4-triazin-3-amine
N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(3-hydroxyphenyl)-4-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-4-oxobutanamide
ethyl 4-[1-(3-phenylpropyl)piperidin-3-yl]piperazine-1-carboxylate
1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(2R,6R)-4-cyclohexyl-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4,6,7-trimethyl-2-{4-[4-(1H-pyrazol-1-yl)butan-2-yl]-1,4-diazepan-1-yl}quinazoline
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}propanamide
1-benzyl-8-(2,3-dihydro-1H-inden-2-yl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cyclohexyl-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-[4-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]ethan-1-one
(2R,3S,6R)-3-(2-methoxyphenyl)-5-[3-(1H-pyrazol-1-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{2-[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
4-(4-ethoxy-3-methylphenyl)-1-[4-(1H-1,2,3,4-tetrazol-5-yl)piperidin-1-yl]butan-1-one
N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-cyclopropylacetamide
N-[2-(2-hydroxyethoxy)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
3,5,7-trimethyl-N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]-1H-indole-2-carboxamide
methyl (2S,4S,5R)-5-(4-chlorophenyl)-1,2-dimethyl-4-(piperidine-1-carbonyl)pyrrolidine-2-carboxylate
N,4-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1,3-thiazol-2-amine
(1S,5R)-6-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
2-(3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
N-[2-(dimethylamino)ethyl]-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine