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3-{[4-(oxan-4-ylmethyl)-3-oxo-6-(pyridin-2-ylmethoxy)-1,4-diazepan-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-[(2,4-dimethoxyphenyl)methyl]-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-ethyl-5-[(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)methyl]pyrimidin-2-amine
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
1-(2-methanesulfonamidoacetyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
4-[4-(4-acetylpiperazine-1-carbonyl)piperidin-1-yl]-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[3-(1H-indol-1-yl)propyl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
methyl 3-(2-chlorobenzenesulfonamido)-5-{[(1,3-dimethyl-1H-pyrazol-5-yl)formamido]methyl}benzoate
3-[(3R,4S)-1-(benzylcarbamoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
11-methyl-4-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-chloro-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}benzene-1-sulfonamide
N-(1-hydroxy-3-methylbutan-2-yl)-5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
5-[(4-benzylpiperidin-1-yl)methyl]-N-[(1-ethylpyrrolidin-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
1-(dimethyl-1,3-thiazole-5-carbonyl)-4-(4-fluorophenyl)-1,4-diazepane
1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
7-(2-methoxyacetamido)-1-methyl-2-phenyl-N-[1-(thiophen-2-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
3-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-methylurea
9-(dimethyl-1,3-oxazole-5-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}adamantan-1-amine
methyl N-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamate
2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(propan-2-ylsulfanyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-hydroxybutanamide
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]furan-2-carboxamide
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
5-(2-phenylethyl)-5-(piperidin-4-yl)-3-(pyridin-3-ylmethyl)imidazolidine-2,4-dione
8-methoxy-N-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
diethyl({[3-(2-ethylpyrrolidine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
methyl 4-{4-[2-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)ethyl]piperidin-1-yl}pentanoate
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
3-ethyl-1-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-1-methylurea
(benzylsulfamoyl)({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl})amine
4-[(furan-2-ylmethyl)amino]-5-methyl-N-[3-(pyridin-4-yl)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
3-(4-fluorophenyl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
9-(3-chlorobenzenesulfonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
N,N-dimethyl-7-(propane-1-sulfonyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(3-fluorophenyl)-1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
N-ethyl-4-[3-(1-methylpiperidin-2-yl)propanamido]piperidine-1-carboxamide
2-(2-hydroxyethyl)-8-[4-(methylsulfanyl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[(4aR,8aR)-7-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
methyl 8-[(5-acetamidothiophen-2-yl)methyl]-1-[(3-methoxyphenyl)methoxy]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
6-(2,5-dimethylfuran-3-yl)-N-(3-hydroxypropyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-phenylethan-1-one
N-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1-(thian-4-yl)piperidin-4-amine
6-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
4-[2-(2,5-dimethylphenoxy)propanoyl]-1-(4-methylphenyl)piperazin-2-one
2-tert-butyl-6-[2-(2-ethoxyethoxy)benzoyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine