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4-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}-1-(propan-2-yl)-1H-pyrazole
6-{1-[3-(2-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}pyrimidin-4-ol
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[1-(2-methoxyphenyl)propan-2-yl]-N-methylacetamide
3-(4-chlorophenyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-phenylpropanamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-3-yl]-1H-1,2,4-triazole-5-carboxamide
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-phenylpiperidine-4-carbonitrile
1-(4-methoxyphenyl)-6,6-dimethyl-N-[(2-methyl-1H-imidazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[(3S,4R)-3-benzyl-1-methylpiperidin-4-yl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
1-(3-methylpyridin-2-yl)-4-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)piperazine
(3S,4S)-4-(azocan-1-yl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidin-3-ol
2-butyl-8-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[2-(dimethylamino)ethyl]-9-(4,6-dimethylpyrimidin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-(1-{1-[(2S)-1-acetylpyrrolidine-2-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(3-fluorophenyl)urea
(3E)-1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pent-3-en-1-one
2-{2-[(dimethylamino)methyl]-4-(pyrimidin-2-yl)phenoxy}-N-{[4-(trifluoromethyl)phenyl]methyl}acetamide
1-{[4-(4-chlorophenyl)-4H-1,2,4-triazol-3-yl]methyl}-4-(2,3-dimethylphenyl)piperazine
3-butyl-4-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-1-methylpiperazin-2-one
1-{4-[7-(methylsulfanyl)-3-({[(3,4,5-trimethoxyphenyl)methyl]amino}methyl)quinolin-2-yl]piperazin-1-yl}ethan-1-one
1-methanesulfonyl-4-(2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenoxy)piperidine
1-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1H-1,2,4-triazol-5-yl]piperidine
3-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
[1-(2-benzyl-1,3-thiazole-4-carbonyl)-2,5-dihydro-1H-pyrrol-2-yl]methanol
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-5-methylpiperidin-2-one
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-(pyrazin-2-yl)propanamide
N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
1-methyl-1'-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
2-[({1-[(4-methanesulfonylphenyl)methyl]piperidin-3-yl}oxy)methyl]pyridine
9-methoxy-7-(3-methoxyphenyl)-4-[(5-methylfuran-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(4-hydroxyazepan-4-yl)methyl]-3-(pyridin-2-yl)propanamide
3-{[(1-methyl-1H-imidazol-2-yl)methyl]sulfamoyl}-N-(pyridin-3-yl)benzamide
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
8-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-[2-methyl-2-(morpholin-4-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
methyl 2-[3-oxo-4-(pyrimidin-5-ylmethyl)-3,4-dihydro-2H-1,4-benzoxazin-2-yl]acetate
ethyl 3-[(3-chlorophenyl)methyl]-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine-3-carboxylate
methyl 5-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-5-oxopentanoate
(1R,2S,9R)-11-(4-aminopyrimidin-2-yl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
7-(2-phenylethyl)-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-{2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethoxy}-4-methyl-1,2,5-oxadiazole
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2,5,6-trimethylpyrimidin-4-amine
(3R,4R)-1-(4-chloro-2-fluorobenzoyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-{4-[5-(2,6-dimethylpyrimidin-4-yl)-1,2,4-oxadiazol-3-yl]phenyl}ethan-1-ol
2-{2,8-diazaspiro[4.5]decan-2-yl}-6-methylpyridine-3-carboxylic acid
2-{[(1-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
5-{4-hydroxy-1-[(4-methylphenyl)methyl]piperidin-4-yl}-N-(thiophen-2-ylmethyl)-1-benzofuran-2-carboxamide
(3R,4R)-1-[(4-methoxypiperidin-1-yl)sulfonyl]-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide