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6-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidine-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
8-(6-aminopyrimidin-4-yl)-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
(2S)-N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-2-acetamidopropanamide
4-(1-methylpiperidin-4-yl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(1,3-benzoxazol-2-yl)ethyl]-1-[4-(furan-2-yl)phenyl]piperidin-4-amine
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
2-{[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
(1S,5R)-3-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(5-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
4-(3-chloro-5-fluoro-4-methoxyphenyl)-1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1H-1,2,3-triazole
5-[1-(cyclohexylmethyl)-4-hydroxypiperidin-4-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
8-(cyclohexylcarbamoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[1-(pyridin-2-yl)propyl]amine
(3-{2-[(dimethylamino)methyl]phenoxy}phenyl)methanol
5-(1-benzothiophen-2-yl)pyrimidin-2-amine
5-{2-[4-(3-chlorophenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
5-(2-fluorophenyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1,2,4-triazin-3-amine
N,N-dimethyl-3-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanamide
2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}thiophen-3-amine
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-3,3,3-trifluoropropan-1-one
N2,N2-dimethyl-N5-[(2-propylpyrimidin-5-yl)methyl]-5,6,7,8-tetrahydroquinazoline-2,5-diamine
2-{5-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}pyridine
2-[(isoquinolin-5-yloxy)methyl]-N-[(1R,2S)-2-phenylcyclopropyl]-1,3-oxazole-4-carboxamide
1-{1-[2-(ethylamino)pyrimidine-5-carbonyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-[4-(3-hydroxyphenyl)piperazine-1-carbonyl]-1-methylpiperidin-4-ol
1-(5-chloro-2-methoxybenzoyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
3-methyl-N-[(3R,4S)-1-[(methylcarbamoyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-1-propyl-1H-pyrazole-4-carboxamide
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-[5-(4-chlorophenyl)-1H-pyrrol-2-yl]-1-[(3S)-3-(dimethylamino)azepan-1-yl]propan-1-one
(2S,4R)-4-amino-1-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-(3-fluorophenyl)-3-oxopiperazine-1-carboxamide
5-(1-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}pyrrolidin-2-yl)thiophene-2-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-1-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
8-(1,4-dithiepan-6-yl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
6-{[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl})(pyridin-4-ylmethyl)amine
2-(3-{[1-ethyl-3-(3-fluoro-4-methylphenyl)-2-oxo-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-6-yl]methyl}-1H-indol-1-yl)acetamide
3-hydroxy-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-one
4-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-4-yl}pyridine
2-(1,3-thiazol-2-yl)-2,8-diazaspiro[4.5]decane
4-(4-chlorophenoxy)-1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidine-4-carboxylic acid
2-[methyl(phenyl)amino]-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-(3,5-dimethoxyphenyl)-2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]acetamide
2,5-dimethyl-3-(3-{1-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrazine
4-[2-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]-1-(propan-2-yl)-1H-pyrazole
8-[2-(4-fluoro-2-methylphenyl)acetyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(3-hydroxypropyl)-1-[5-(4-methylphenyl)-1H-pyrazole-3-carbonyl]piperidine-3-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione