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N-(2,3-dihydro-1H-inden-2-yl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}-2-[3-(methylcarbamoyl)phenyl]acetic acid
5-{pyrazolo[1,5-a]pyridin-7-yl}pyrimidin-2-amine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(3-hydroxy-3-methylbutyl)-N-methylacetamide
N-{2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]thiophen-3-yl}acetamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[2-(methylsulfanyl)benzoyl]pyrrolidin-3-yl]methanol
8-[3-(2-methyl-1H-indol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
N'-cyclopentyl-N-(cyclopropylmethyl)-N-(oxolan-2-ylmethyl)butanediamide
N-ethyl-5-methyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
(1R,2S)-N-(prop-2-en-1-yl)-2-(4-propylpiperazine-1-carbonyl)cyclohexane-1-carboxamide
1-[2-(4-chlorophenyl)ethyl]-N-methyl-6-oxo-N-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
3-{2-[2-(1-benzofuran-2-yl)-1H-imidazol-1-yl]ethyl}-5-(oxolan-2-yl)-1,2,4-oxadiazole
N-(1-benzoylpiperidin-3-yl)-3-(1-methyl-1H-pyrazol-5-yl)propanamide
{4-[(3-chloro-4-propoxyphenyl)methyl]-1-methylpiperazin-2-yl}methanol
3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methyl-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
N-[(3R,4S)-4-cyclopropyl-1-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]pyrrolidin-3-yl]cyclopentanecarboxamide
7-chloro-2-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
1-(2,3-dihydro-1H-inden-2-yl)-4-(pyrimidin-2-yl)-1,4-diazepane-6-carboxylic acid
N5-cyclopropyl-N6-(2,2-dimethyloxan-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-{3-[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]phenyl}-N-methylpropanamide
4-(3-cyclohexylpyrrolidin-1-yl)-1-ethylpiperidine
3-({[4-(pyridin-2-yl)pyrimidin-2-yl]amino}methyl)-1λ6-thiolane-1,1-dione
N-{5-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-2-methylphenyl}cyclopentanecarboxamide
2-methyl-N-[1-(thiophen-2-yl)butyl]pyrido[2,3-d]pyrimidin-4-amine
methyl 6-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-3-[2-(2-methylphenyl)acetamido]thieno[2,3-b]pyridine-2-carboxylate
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-benzyl-1,3-thiazole-4-carboxamide
4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-2-(3-fluorophenoxymethyl)-1,3-oxazole
4-[2-(dimethylamino)acetamido]-N-(1-phenylbutyl)benzamide
1'-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(3-methylbutyl)propanamide
2-{4-[(6-hydroxy-1,4-oxazepan-6-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
6-[4-(1-cyano-1-methylethyl)phenyl]-N-methylpyridine-2-carboxamide
8-[3-(3,4-dimethoxyphenyl)propanoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
7-(3-chlorophenyl)-4-(2-fluorobenzoyl)-9-(pyridin-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(5-methylfuran-2-yl)-N-{2-[6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidin-4-yl]ethyl}-1H-pyrazole-5-carboxamide
(2S,4R)-N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
8-[(5-chloro-2-hydroxyphenyl)methyl]-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)pyridine-2-carboxylic acid
5-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-2-(piperidin-1-yl)pyrimidine
N-[2-(piperazin-1-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
5-methoxy-4-oxo-N-(2,2,2-trifluoroethyl)-1,4-dihydropyridine-2-carboxamide
8-[(3-chloro-4-fluorophenyl)carbamoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-methoxy-6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidine
N-(oxolan-2-ylmethyl)-N-propyl-1H-1,2,4-triazole-5-carboxamide
(1S,5R)-3-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
{3-[(3-methoxyphenyl)methyl]-1-(9H-purin-6-yl)piperidin-3-yl}methanol
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-[3-(2-methylphenoxy)azetidin-1-yl]propan-1-one
1-{[1-(2,3-dihydro-1H-inden-5-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazole
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-(1H-indole-6-carbonyl)pyrrolidin-3-yl]methanol
4-[4-(2-ethoxyphenyl)piperazin-1-yl]-6-(methoxymethyl)pyrimidine