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1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(3-methylthiophene-2-carbonyl)piperidine
1-[2-(4-fluorophenyl)piperidin-1-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
2-{[ethyl(oxan-4-ylmethyl)amino]methyl}-6-methoxyphenol
5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]pyridine-2-carbonitrile
4-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]-1,2-dihydroisoquinolin-1-one
4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-(propan-2-yl)piperidine
5-methyl-3-(3-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)-1,2,4-oxadiazole
N-{[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-fluorobenzamide
2-(methoxymethyl)-6-methyl-N-[2-(morpholin-4-yl)ethyl]-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butan-1-one
1-[(3-methylpyridin-2-yl)methyl]-4-[2-(methylsulfanyl)benzoyl]piperazine
4-(1-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)-1-(propan-2-yl)piperidine
2-(3-methoxypropyl)-8-(3-methyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-[(6-ethoxypyridin-3-yl)methyl]-2-(pyridin-3-yl)morpholine
1-(2-{[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]methyl}phenyl)-1H-1,2,4-triazole
N-cyclohexyl-1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-4-carboxamide
N-[3-({[3-(pyridin-4-yl)propyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
3-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-1-[2-methyl-3-(1H-pyrrol-1-yl)phenyl]urea
1-(2-methoxyethyl)-4-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]pyrrolidin-2-one
4-[(4aR,8aR)-4a-hydroxy-7-methanesulfonyl-decahydro-2,7-naphthyridin-2-yl]-1-phenylbutan-1-one
1-[(4-fluorophenyl)methyl]-4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
2-(1-benzofuran-2-yl)-4,6-dimethylpyridine-3-carboxamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-3-(2-oxopyrrolidin-1-yl)propanamide
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
4-[1-(2-phenoxyethyl)-1H-1,2,3-triazol-4-yl]-1-(propan-2-yl)piperidine
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-(benzyloxy)ethan-1-one
N-[(4-fluorophenyl)methyl]-4-(5-oxo-1,4-diazepan-1-yl)pyridine-2-carboxamide
N-(4-{4-[(1,4-dioxan-2-ylmethyl)(methyl)amino]piperidin-1-yl}phenyl)-2,4-dimethylbenzamide
N-[(4-fluorophenyl)methyl]-2-(4-propanoylphenoxy)-N-(pyridin-4-ylmethyl)acetamide
(1R,5R)-6-propyl-3-{thieno[2,3-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonane
1-(1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)-3-propylpiperidine-3-carboxylic acid
N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
4-[4-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)piperazin-1-yl]benzoic acid
6-[(2R,3R)-3-[ethyl(methyl)amino]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]pyridine-3-carboxamide
N-(9H-fluoren-9-yl)-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
8-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{2-amino-4-[(2-methylprop-2-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(piperazin-1-yl)ethan-1-one
8-[(5-chloro-2,4-dimethoxyphenyl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
4-[(2-fluorophenyl)methyl]-1-[4-(1H-pyrazol-1-yl)benzoyl]-1,4-diazepan-5-one
4-benzyl-3-ethyl-1-(1H-indazole-3-carbonyl)-1,4-diazepan-5-one
N-butyl-2-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-imidazole-4-carboxamide
1-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-1H-1,2,3-triazole
[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropylimidazo[1,2-a]pyridine-6-carboxamide
4-[4-(3-chlorophenyl)-1H-imidazol-2-yl]-1-cyclopropylpyrrolidin-2-one
1-cyclopentyl-N-(3-methylbutyl)-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
(4aS,7aR)-1-[(2,6-dimethoxyphenyl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S)-2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-4-(methylsulfanyl)butan-1-ol