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N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,3-difluorobenzamide
N-(2,3-dihydroxypropyl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(oxan-4-yl)propanamide
N-ethyl-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(pyridin-4-ylmethyl)benzamide
1-(2-methylpyridin-4-yl)-4-[3-(methylsulfanyl)butyl]-1,4-diazepane
2-(2-tert-butylpyrimidin-5-yl)-7-fluoro-N-methyl-N-(propan-2-yl)quinoline-4-carboxamide
3-{[1-(2-ethylbenzoyl)piperidin-4-yl]methyl}benzoic acid
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-3,5-dimethyl-1-benzofuran-2-carboxamide
(1-{[1-(2,3-dimethylquinoxaline-6-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-2-yl}methanol
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[(3R,4R)-3-hydroxy-1-(quinolin-4-ylmethyl)piperidin-4-yl]pyridine-3-carboxamide
4-[(3Z)-hex-3-en-1-yl]-1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-1,2,3-triazole
7-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-N,N-dimethyl-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(1-benzofuran-2-yl)-2-{methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}acetic acid
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
1-[1-(5-cyanopyridin-2-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
[1-(1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)piperidin-4-yl]methanol
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-(pyridine-2-carbonyl)piperazin-2-yl}ethan-1-ol
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(1,3-oxazole-5-carbonyl)piperidin-3-yl]propanamide
3-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)piperidin-4-yl]-1,3-oxazolidin-2-one
2-methyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,3-benzoxazole-6-carboxamide
5-[1-(2-methoxyethyl)-1H-pyrazol-3-yl]-4-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,3-thiazol-2-amine
2-(2-chlorophenyl)-3-methyl-N-(propan-2-yl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-tert-butyl-3-(thiophen-2-ylmethyl)-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
8-[(2-cyclohexylpyrimidin-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5-[(2E)-3-phenylprop-2-enoyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-{4-[(6-fluoroquinolin-2-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-ethyl-7-methoxy-4-(2-methylbutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3R,4S)-1-{5-[(diethylamino)methyl]-2-phenylfuran-3-carbonyl}-3,4-dimethylpiperidin-4-ol
methyl 3-[3-(morpholin-4-ylmethyl)phenyl]benzoate
3-{2-[4-(4-fluorophenyl)piperazin-1-yl]-2-oxoethyl}-4-(propan-2-yl)piperazin-2-one
N-(4-{[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]methyl}phenyl)acetamide
1-[(4-fluorophenyl)methyl]-5-[3-(methylsulfanyl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
6,7-dimethoxy-2-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
N-ethyl-5-[4-(4-methylbenzenesulfonyl)piperazine-1-carbonyl]pyrimidin-2-amine
methyl (2S,4R)-1-methyl-4-[3-(5-methyl-1,2,4-oxadiazol-3-yl)benzamido]pyrrolidine-2-carboxylate
(3R,4S)-1-[(4-methylpiperidin-1-yl)sulfonyl]-4-propylpyrrolidin-3-amine
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-methyl-N-[3-(morpholin-4-yl)propyl]-1,2-oxazole-3-carboxamide
(2S)-2-{[(4-hydroxy-6-methylquinolin-2-yl)methyl]amino}-4-methylpentanamide
methyl (2R)-2-[(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazol-4-yl)formamido]propanoate
2-(furan-2-yl)-1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidine
(3R,4S)-4-cyclopropyl-1-[(1-methyl-1H-1,2,3-benzotriazol-4-yl)sulfonyl]pyrrolidin-3-amine
1-{[4-(methylsulfanyl)phenyl]methyl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
(1S,5R)-6-(cyclobutylmethyl)-3-(2-ethylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-hydroxy-N-({1-[(2E)-2-methylpent-2-en-1-yl]piperidin-3-yl}methyl)-4-oxo-4H-pyran-2-carboxamide
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
1-propyl-5-[4-(1H-1,2,4-triazol-3-yl)phenyl]-1H-1,2,4-triazole