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N-ethyl-4-{[2-(pyrazin-2-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
N1,N1-dimethyl-N3-{2-[methyl(phenyl)amino]ethyl}piperidine-1,3-dicarboxamide
3-(dimethyl-1,2-oxazole-4-carbonyl)-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-{2-methylimidazo[1,2-a]pyridin-3-yl}-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide
3-methanesulfonamido-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)propanamide
3-[(2R,3R,6R)-5-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
4-[1-(1-benzylpiperidin-4-yl)piperidine-3-carbonyl]piperazin-2-one
3-methyl-N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}-1H-pyrazole-5-carboxamide
2-(3-phenylpropyl)-8-(pyridine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(3aS,6aS)-2-(cyclopropylmethyl)-1-oxo-5-{thieno[2,3-d]pyrimidin-4-yl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-[3-(3,5-dimethylphenyl)propanoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-{[3-(4-methoxyphenoxy)phenyl]methyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
2-[4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
1-(6-hydroxy-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-1,4-diazepan-1-yl)ethan-1-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[3-(2-hydroxyphenyl)propyl]acetamide
3-chloro-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
4-benzyl-3-ethyl-1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-1,4-diazepan-5-one
{1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-3-(3-methoxypropyl)piperidin-3-yl}methanol
(1S,4S)-2-(3,4-difluorophenyl)-5-(2,6-dimethoxybenzoyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
5-ethyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1,3-oxazole-4-carboxamide
methyl 4-{[4-(pyridin-4-yl)piperidine-1-carbonyl]amino}benzoate
3-[1-(2-methoxy-2-methylpropyl)-1H-imidazol-2-yl]quinolin-7-ol
N-benzyl-N,1-dimethyl-5-{methyl[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(3R,4S)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3-hydroxypropanamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-methyl-N-(oxan-4-yl)acetamide
3-(cyclopropylmethyl)-1-(4-fluorobenzoyl)piperidine-3-carboxylic acid
N3-ethyl-N5-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(3R,5S)-1-(2-methoxyethyl)-5-(methylcarbamoyl)pyrrolidin-3-yl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
(2S,4R)-N-methyl-1-(propan-2-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
N-({1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
N-[(5-methoxy-1H-indol-2-yl)methyl]-4,6-dimethylpyrimidin-2-amine
8-(9H-fluoren-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
2-{3-[(dimethylamino)methyl]phenyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{3-[(diethylamino)methyl]phenyl}-4-(pyridin-3-yl)piperazine-1-carboxamide
5-[(3-fluorophenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
3-hydroxy-1-(2-phenylethyl)-3-[(4-phenylpiperazin-1-yl)methyl]piperidin-2-one
1-methyl-4-{5-[(1-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}piperazine
2-acetyl-8-(5-fluoro-2-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-fluoro-N-({1-[2-(methylsulfanyl)acetyl]piperidin-3-yl}methyl)benzamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}propanamide
4-[4-(azonane-1-carbonyl)phenyl]-2-methylbutan-2-ol
1-(furan-3-ylmethyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-{[methyl({4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl})amino]methyl}-3,4-dihydroquinazolin-4-one
1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methylphenoxy)piperidine
1-{[1-tert-butyl-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1S,6R)-9-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-3,9-diazabicyclo[4.2.1]nonane
(3R,4R)-1-[(8-chloroquinolin-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-ol
8-[(2-ethylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one