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3-[2-(dimethylamino)ethyl]-5-[1-(2,4-dimethylbenzoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
N-cyclohexyl-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
(2S)-N-[4-(3-methoxyphenyl)phenyl]-1-[2-(4H-1,2,4-triazol-4-yl)ethyl]pyrrolidine-2-carboxamide
4-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)morpholine
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
3-(1H-imidazol-1-ylmethyl)-1-(2-phenylethyl)piperidine
3-(2-methylpropyl)-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1,2-oxazole-5-carboxamide
2-{[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,3-benzothiazole
7-[1-(2-fluorophenyl)piperidin-4-yl]-2-oxa-7-azaspiro[4.5]decan-8-one
4-ethyl-3-(1-{7-methyl-2-oxo-1H,2H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-benzyl-N,1-bis(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
2-(2,4-difluorophenoxy)-1-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]ethan-1-one
N-[3-(2-fluorophenyl)propyl]-1-methylazepane-2-carboxamide
2-{N-[(2-methoxyphenyl)methyl]-1-(2-methyl-1-benzofuran-5-yl)formamido}acetic acid
5-ethyl-N-methyl-N-(quinoxalin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(3,3-dimethyl-2-oxobutyl)benzamide
4-methoxy-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
2-methyl-8-(5-phenyl-1H-pyrrole-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-{[1-(2-hydroxybutyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}methanesulfonamide
3-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-ylmethyl]benzonitrile
1-[3-(hydroxymethyl)-4-methylpiperazin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-1H-pyrazole-4-carbonyl)-4-methylpiperazine
5-ethyl-N-{[1-(2-phenylethyl)piperidin-4-yl]methyl}-1,3,4-oxadiazol-2-amine
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
1-{1-[6-(hydroxymethyl)pyridine-2-carbonyl]-4-phenylpiperidin-4-yl}ethan-1-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N,1-dimethyl-1H-indole-2-carboxamide
(3R,4S)-1-(3-fluoropyridin-2-yl)-3,4-dimethylpiperidin-4-ol
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-[2-(1H-imidazol-1-yl)ethyl]acetamide
4-{6-[1-(3-ethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]pyrimidin-4-yl}morpholine
1-[(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2-methoxyphenyl)methyl]pyrrolidine
(2Z)-N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-fluoro-3-phenylprop-2-enamide
(3R,5S)-N-[2-(benzylsulfanyl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-5-[(methylsulfanyl)methyl]furan-2-carboxamide
2-(3-{3-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]phenyl}-1H-pyrazol-1-yl)ethan-1-ol
4-[(4aS,8aS)-7-cyclopentanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridine-2-carbonyl]benzonitrile
methyl 4-(5-{[2-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
4-(carbamoylmethoxy)-N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)benzamide
8-cyclobutanecarbonyl-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethyl-1,3-thiazole-4-carboxamide
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-ethyl-1-(5-methanesulfonyl-2-methylphenyl)urea
11-[4-methoxy-3-(prop-2-en-1-yl)phenyl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
(2S)-2-[(1-benzyl-1H-pyrazol-4-yl)formamido]-3-(4-hydroxyphenyl)propanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-(methoxymethyl)-N-(pentan-3-yl)cyclopropane-1-carboxamide
N-[2-(3,5-dimethoxyphenyl)-2-hydroxyethyl]-1-methylpiperidine-4-carboxamide
2-{2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethoxy}ethan-1-ol
4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1,4-oxazepan-6-ol
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
N-[(2,3-difluoro-4-methylphenyl)methyl]-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
5-(3-acetylphenoxymethyl)-N-(2,3-dihydroxypropyl)-N-methyl-1H-pyrazole-3-carboxamide