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2-(4-acetylphenoxy)-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}acetamide
1-[2-(1H-pyrazol-1-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N1-[4-(3-methoxyphenoxy)phenyl]-N2-methylpyrrolidine-1,2-dicarboxamide
2-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-4-(pyrimidin-5-yl)phenol
1-(3,3-dimethylbutanoyl)-4-(2-methylpropyl)-1,4-diazepan-5-one
methyl({[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})(2-methylpropyl)amine
{1-[1-(1-methyl-1H-imidazole-2-carbonyl)piperidin-4-yl]piperidin-3-yl}methanol
6-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-9H-purin-2-amine
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-amine
2-(ethylamino)-N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}pyrimidine-5-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
3-(1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)propan-1-ol
5-{[benzyl(methyl)amino]methyl}-N-(1-hydroxy-3-methylbutan-2-yl)-1,2-oxazole-3-carboxamide
1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
4-hydroxy-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide
ethyl 1-[5-(methoxymethyl)furan-2-carbonyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
2-({1-[(3-acetylphenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
ethyl 1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-4-(2-methoxyethyl)piperidine-4-carboxylate
1-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-4-methyl-1,4-diazepane
1-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-3-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]urea
N-[(2,3-difluorophenyl)methyl]-1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-amine
1-ethyl-5-[3-methyl-1-(4-methylphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-imidazole
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(thiophen-2-ylsulfanyl)pyrimidin-2-amine
(4aS,7aR)-1-(1-aminocyclopropanecarbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,4R)-4-cyclopropyl-3-methyl-1-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidin-4-ol
{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl){[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}amine
(3S)-3-ethyl-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}morpholine
N-(2,6-difluorophenyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecane-11-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
4-phenoxy-1-[3-(1H-pyrazol-1-yl)propanoyl]piperidine-4-carboxylic acid
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
3-(3,5-dimethoxyphenyl)imidazo[1,2-b]pyridazine
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[4-(piperidin-1-yl)benzoyl]piperidin-3-amine
2-(ethylsulfanyl)-1-[1-(hydroxymethyl)-9-[(1-methyl-1H-imidazol-5-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
2-ethyl-9-[(2-fluorophenyl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
1-{3-[(E)-2-phenylethenyl]phenyl}piperazine
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]piperidine-4-carboxamide
2-methoxyethyl 2-(2-phenylethyl)piperidine-1-carboxylate
1-(2-{[(1-phenyl-1H-pyrazol-5-yl)carbamoyl]amino}ethyl)piperidine-3-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(1H-1,2,3-triazol-1-yl)ethan-1-one
N4-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-6-methylpyrimidine-2,4-diamine
2-(2-fluorophenoxymethyl)-N-methyl-N-(1-methylpiperidin-4-yl)-1,3-oxazole-4-carboxamide
2-[1-(propan-2-yl)piperidin-4-yl]-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}acetamide
9-[2-(2-methoxyethoxy)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
N-(furan-2-ylmethyl)-3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-(3,4-dichlorophenyl)-4-(2-methoxypyridine-3-carbonyl)morpholine