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(3S,4R)-4-methyl-1-(1-methyl-1H-indole-3-carbonyl)piperidine-3,4-diol
N-(butan-2-yl)-4-[(1H-indol-4-ylmethyl)sulfamoyl]benzamide
1-(1H-1,3-benzodiazol-2-ylmethyl)-4-phenylpiperidine-4-carbonitrile
methyl 3-[cyclopentyl({[4-methoxy-3-(propan-2-yloxy)phenyl]methyl})sulfamoyl]thiophene-2-carboxylate
1-{2-oxo-2-[3-(4-phenoxybenzoyl)piperidin-1-yl]ethyl}piperidin-2-one
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(4-propanoylphenoxy)acetamide
2-{[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amino}-N-(pyrazin-2-yl)acetamide
5-methyl-3-(2-{2-oxa-7-azaspiro[4.5]decan-7-yl}-2-oxoethyl)-2,3-dihydro-1,3-benzoxazol-2-one
(4aR,7aS)-1-ethyl-4-{[3-(trifluoromethoxy)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2-methoxyethyl)-8-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}pyridin-2-amine
N-{2-[(4-ethyl-5-methylpyrimidin-2-yl)amino]ethyl}-N-methylmethanesulfonamide
8-[(2-aminopyridin-3-yl)methyl]-2-[(3,4-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
5-methoxy-3-methyl-2-{[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]methyl}-1H-indole
2-(cyclopropylmethyl)-9-{2-[methyl(phenyl)amino]acetyl}-2,9-diazaspiro[5.5]undecan-3-one
1-(2,2-dimethylpropyl)-3-hydroxy-3-[(4-hydroxypiperidin-1-yl)methyl]piperidin-2-one
[3-(5-methyl-1,2-oxazole-3-carbonyl)-9-[3-(methylsulfanyl)propyl]-3,9-diazaspiro[5.5]undecan-1-yl]methanol
1-{3-[(3-fluorophenyl)methoxy]benzoyl}-3,4,4-trimethylpyrrolidin-3-ol
2-cyclopropyl-N-[(4-phenyloxan-4-yl)methyl]-1,3-benzoxazole-6-carboxamide
4-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)thiomorpholine
1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,3-triazole
(2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}pyridin-4-yl)methanol
ethyl 4-(2-phenylethyl)piperidine-4-carboxylate
3,3,3-trifluoro-N-[(3R,4S)-1-(2-methoxyethyl)-4-(propan-2-yl)pyrrolidin-3-yl]propanamide
3-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-1-ethyl-1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]urea
methyl 1-(2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetyl)piperidine-4-carboxylate
N,2,5-trimethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}furan-3-carboxamide
1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-phenyl-2-(phenylamino)propan-1-one
N-{2-[3-(4-tert-butylbenzoyl)piperidin-1-yl]-2-oxoethyl}acetamide
1-(2-fluorophenyl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclopropane-1-carboxamide
N-(4-chloro-2-fluorophenyl)-2-{[2-(pyridin-4-ylformamido)ethyl]amino}acetamide
5-{2-[4-(4-chloro-1-methyl-1H-indazol-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,3,4-thiadiazol-2-amine
4-cyclohexyl-3-[(4-hydroxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[2-(morpholin-4-ylmethyl)phenyl]-1-[2-(pyridin-3-yloxy)propyl]urea
N-[3-(4-hydroxyphenyl)propyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)propanamide
(2R,6S)-4-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2,6-dimethylmorpholine
2-oxo-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)-1-oxaspiro[4.4]nonane-4-carboxamide
N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)thiophene-2-carboxamide
methyl 2-[(2,3-dimethylphenyl)sulfamoyl]-6-[(2-hydroxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(dimethylamino)-2-(3-methylphenyl)-N-(quinolin-4-ylmethyl)acetamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(2-methoxy-3-methylbenzoyl)pyrrolidin-3-yl]methanol
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-benzyl-N3-[1-(4-fluorophenyl)ethyl]-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[3-(furan-2-yl)phenyl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine-4-carboxamide
N4-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylisoquinoline-5-carboxamide
3-(2-methoxyphenoxy)-1-(5-propylthiophene-3-carbonyl)azetidine
3-{1-[3-(3,5-dimethylphenyl)propanoyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)-1-methyl-1,2,3,4-tetrahydroquinolin-2-one