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1-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-3-ethylpiperidine-3-carboxylic acid
6-tert-butyl-2-(2-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-[2-(4-acetyl-1,4-diazepan-1-yl)-2-oxoethyl]-4-(cyclohexylmethyl)piperazin-2-one
1-[3-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
2-{1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
1-methyl-2-(2-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)-1H-1,3-benzodiazole
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[(4-hydroxyquinolin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidin-2-one
3-{5-[2-(1H-pyrrol-1-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-[4-(propan-2-yl)morpholin-2-yl]-1-[4-(pyridin-3-ylmethyl)piperazin-1-yl]ethan-1-one
2-[(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)methyl]benzoic acid
N-[4-({[2-(2-ethoxyphenoxy)ethyl](methyl)amino}methyl)phenyl]acetamide
2-({[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)amino)-1-phenylethan-1-ol
3-[1-(naphthalene-1-sulfonyl)azetidin-3-yl]pyridine
N,N-dimethyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidin-4-amine
(1R,2R,6S,7S)-4-[4-(1H-pyrazol-3-yl)benzoyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)-1,2,3-thiadiazole-4-carboxamide
N-[2-(4-methylphenyl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
3-[(3R,4S)-1-[3-(2,3-dihydro-1H-isoindol-2-yl)propanoyl]-4-(dimethylamino)piperidin-3-yl]propanoic acid
2-cyclobutyl-5-(2-methoxyacetamido)-N,1-dimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
1-cycloheptyl-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
N-(1-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
3-{1-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]piperidin-3-yl}-N-(2-fluorophenyl)propanamide
5-[5-(dimethylcarbamoyl)furan-2-yl]thiophene-2-carboxylic acid
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(pyrrolidine-2-carbonyl)piperidine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-methanesulfonamidopropanamide
4,4-difluoro-1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
[1-(3-methoxypropyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
N-(oxolan-2-ylmethyl)-N-({4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-3-(trifluoromethyl)benzene-1-sulfonamide
2-(3-{[ethyl(oxan-2-ylmethyl)amino]methyl}phenoxy)acetamide
(2S,4S)-4-amino-1-{[4-methoxy-3-(prop-2-en-1-yl)phenyl]methyl}-N-methylpyrrolidine-2-carboxamide
(4-{[1-(2H-1,3-benzodioxol-5-ylmethyl)pyrrolidin-3-yl]methyl}phenyl)methanol
3-{4-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
(1S,3R)-3-amino-N-[(1-ethyl-1H-indazol-3-yl)methyl]cyclopentane-1-carboxamide
methyl 2-[1-(2-methoxyethyl)-2,4-dioxo-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
(2S,4S)-4-{[(3-methoxyphenyl)methyl]amino}-1-[(2E)-3-phenylprop-2-en-1-yl]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2,8-dimethylquinoline-4-carboxamide
3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-[3-(1H-imidazol-5-yl)phenyl]urea
N-[(3S,4R)-1-(2-methoxyethyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
1-{1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
1-[3-(phenylsulfanyl)propyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
methyl 4-{[1-(3-phenylpropyl)piperidin-3-yl]carbamoyl}butanoate
6,6-dimethyl-1-phenyl-N-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
methyl 4-{[(2-{1-[2-(2-fluorophenyl)ethyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
N-[3-(pyridin-2-yl)propyl]-6-[(quinolin-3-ylmethyl)amino]pyridine-3-carboxamide
1-{[2-(cyclopentyloxy)phenyl]methyl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
N-[(3R,4S)-4-cyclopropyl-1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methanesulfonamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-(piperidin-1-ylmethyl)benzamide