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1-methyl-3-({1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}methyl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(2,6-difluorophenoxymethyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
methyl N-(2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)carbamate
4-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}pyridine
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-methyl-2-(phenylamino)propan-1-one
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-{[1-(methylcarbamoyl)propyl]sulfamoyl}benzamide
N-[3-(2,6-dimethylphenoxy)propyl]-N,5-dimethylpyridine-3-carboxamide
4-(2-methyl-6-propylpyrimidin-4-yl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[2-(pyridine-3-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-4-carboxamide
4-{[1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}benzoic acid
1-{2-[3-(3-chlorobenzoyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
3-(3-fluorophenyl)-4-[2-(methylamino)acetyl]piperazin-2-one
2-(3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl)benzoic acid
7-hydroxy-4-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
N-[(2R,3R)-2-ethoxy-1'-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
1-[(2-fluorophenyl)methyl]-8-(quinolin-6-yl)-1,8-diazaspiro[4.5]decane
1-[3-(methoxymethyl)pyrrolidin-1-yl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethan-1-one
6-methyl-2-(4-{[methyl({[1-(2-methylpropyl)pyrrolidin-3-yl]methyl})amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
ethyl 1-ethyl-5-(1H-indole-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-[(3-methylthiophen-2-yl)methyl]benzamide
(2E)-3-(2,6-difluorophenyl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]prop-2-enamide
8-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-[(3-methylquinoxalin-2-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-3-ol
2-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-cycloheptylpiperidine
2-(4-chlorophenyl)-4-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]morpholine
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]butanamide
(1S,2S)-2-[4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]cyclohexan-1-ol
N-(pyridin-3-ylmethyl)-4-{1H-[1,2,3]triazolo[4,5-b]pyridin-6-yl}-1H-pyrrolo[2,3-b]pyridin-6-amine
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperidine
2-[4-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole
1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-2-{[(2-fluorophenyl)methyl](methyl)amino}ethan-1-one
3-benzyl-5-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
2-{5-[1-(2-chloro-4-fluorophenoxy)ethyl]-3-cyclopentyl-1H-1,2,4-triazol-1-yl}acetic acid
N-{1-[(2-ethylpyrimidin-5-yl)methyl]azepan-4-yl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
(2S,4S)-N,N-diethyl-4-[2-(methylsulfanyl)acetamido]-1-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
3-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-1-(2-phenylphenyl)urea
N-[4-(furan-2-ylmethoxy)phenyl]-3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carboxamide
1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-phenyl-5-(2,4,5-trimethoxyphenyl)-1H-imidazole
ethyl 4-[2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetyl]piperazine-1-carboxylate
2-[(4-chlorophenyl)methyl]-8-(3-fluoropyridin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N-cyclopentyl-3-(1,2-oxazinan-2-yl)-N-(prop-2-en-1-yl)propanamide
1-[(1S,5R)-6-(naphthalene-2-sulfonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-methyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-(thiophen-3-ylmethyl)acetamide
(3aS,6aS)-2-[2-(2-fluorophenyl)acetyl]-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(2,5-dimethylbenzoyl)-2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-cyclopropyl-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[4-(morpholin-4-ylmethyl)phenyl]urea
(2S)-1-(furan-3-ylmethyl)-N-[3-(1H-indol-2-yl)phenyl]pyrrolidine-2-carboxamide
2-{1-[(4-methylphenyl)methyl]-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol