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4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-(thiophen-3-ylmethyl)piperidine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(3-ethyl-1,2-oxazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4,4,4-trifluoro-N-[(4-methylphenyl)(pyridin-4-yl)methyl]butanamide
N-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)oxolane-3-carboxamide
2-methyl-4-(4-{[2-(trifluoromethyl)morpholin-4-yl]methyl}phenyl)butan-2-ol
6-oxo-1-(prop-2-en-1-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]piperidine-3-carboxamide
1-benzyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-pyrazole-4-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-1-(pyrimidin-2-yl)piperidin-4-amine
3-fluoro-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-(1H-1,2,4-triazol-3-yl)benzamide
5-methyl-N-[3-(morpholin-4-yl)propyl]-2-phenylfuran-3-carboxamide
6-{2-amino-4-[(prop-2-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
6-[(3S)-3-hydroxypyrrolidin-1-yl]-N-propylpyridine-3-carboxamide
1-(diphenylmethyl)-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-1H-1,2,3-triazole-4-carboxamide
(3S,9aR)-3-(1H-indol-3-ylmethyl)-8-(thiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(3-{[1-(2-methylfuran-3-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-(2-{7-[(2E)-3-(3-chlorophenyl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methylbenzamide
(7-chloro-5-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-2,3-dihydro-1-benzofuran-2-yl)methanamine
[1-({1-[(6-chloroquinolin-2-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
N-[3-(2-methoxyphenoxy)propyl]-N-methyl-2,3-dihydro-1H-indene-1-carboxamide
ethyl 1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
1-benzyl-4-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1H-pyrazole
(3aS,6aS)-2-cyclohexyl-5-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-(1-methyl-1H-pyrazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(3-benzoylpiperidine-1-carbonyl)pyrazin-2-ol
1-[(2E)-3-phenylprop-2-en-1-yl]-4-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperazine
2-(1-methyl-1H-1,3-benzodiazol-2-yl)-N-(prop-2-en-1-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-{4-[1-methyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]phenyl}pyrrolidin-2-one
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-3-(furan-2-yl)propan-1-one
N-(cyclopropylmethyl)-N-methyl-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
1-{4-[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
[(2S,6S)-4-[(5-fluoro-2-methoxyphenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
(2S,4S,5R)-5-(2,3-difluorophenyl)-1-methyl-4-[methyl(pyridin-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
(2S)-1-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}pyrrolidine-2-carboxamide
N4-[2-(tert-butylsulfanyl)ethyl]-5-ethylpyrimidine-2,4-diamine
4-(2-methyl-1H-imidazol-1-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]butan-1-one
ethyl 1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
2-[1-(cyclohexylmethyl)-4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
(3R,4R)-N-[(2-fluorophenyl)methyl]-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[(3R,4S)-4-(4-methoxyphenyl)-1-methylpyrrolidin-3-yl]acetamide
N-[1-(2-methoxyphenyl)propan-2-yl]-N-methyl-N'-(4-methylphenyl)propanediamide
2-methyl-5-{3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
N-[3-(3-methylphenyl)phenyl]-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-3-carboxamide
3-oxo-N-phenyl-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-{[4-(morpholin-4-yl)phenyl]methyl}propanamide
4-[4-(adamantan-1-yl)piperazine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide