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N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(thiophene-3-carbonyl)piperidine-2-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
methyl (2S)-2-{[6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-3-methylbutanoate
1-({5-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)azepane
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(oxan-2-ylmethyl)-1,2-oxazole-3-carboxamide
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
5-chloro-6-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]pyridine-3-carboxylic acid
N-[1-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-2-carboxamide
(2R,6R)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-{3-[1-tert-butyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]phenoxy}acetamide
2,6-dimethoxy-3-[3-(2-methoxyethyl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]pyridine
2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
N-[(3R,4S)-4-cyclopropyl-1-[2-(morpholin-4-yl)benzoyl]pyrrolidin-3-yl]acetamide
7-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-methyl-6-(2-methylphenyl)-N-(oxan-4-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(isoquinolin-5-ylmethyl)(methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
1-cyclopentyl-4-[4-(naphthalen-2-yl)-1H-pyrazol-5-yl]piperidine
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(3,4-difluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
(1S,4S)-2-(2-chlorophenyl)-5-{[4-(methylsulfanyl)phenyl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
1-cyclobutyl-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
5-(methoxymethyl)-N-[3-(pyrrolidin-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(3-methylphenoxy)-1-{4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
1'-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(1H-1,3-benzodiazol-1-yl)-N-cyclopropyl-N-[(2-methoxyphenyl)methyl]propanamide
2-(2-methyl-1,3-thiazol-4-yl)-1-[3-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-ol
1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
1-(3-ethyl-1H-pyrazole-4-carbonyl)-2-(2-phenylethyl)piperidine
2-methoxy-6-{[(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amino]methyl}phenol
N2-benzyl-6-(2,3-dichlorophenyl)-1,3,5-triazine-2,4-diamine
4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{1-[(2-hydroxy-6-methoxyquinolin-3-yl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-3-(thian-4-yl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(3-methoxypiperidin-1-yl)-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridine
1-{1-[(3-chlorophenyl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine
3-({[1-(methoxymethyl)cyclopentyl]carbamoyl}amino)-2-methyl-N-(2-methylpropyl)benzamide
3-[3-chloro-4-(1H-imidazol-1-yl)phenyl]-1-(piperidin-4-ylmethyl)urea
N-[3-(benzyloxy)phenyl]-2-(2-methoxyethyl)morpholine-4-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
8-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-(1-{7-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-(2-phenoxyethyl)acetamide
1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
(3S,4R)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
3-cyclohexyl-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-1H-pyrazole-4-carboxamide
N-(3-chloro-4-propanamidophenyl)-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanamide
4-ethyl-1-methyl-3-{1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
6-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-3-(3-fluorophenyl)-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-(1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidin-2-yl)pyridine