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4-[4-(1H-indol-4-ylmethyl)piperazin-1-yl]butan-1-ol
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
(3R,4R)-4-(azepan-1-yl)-1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperidin-3-ol
1-tert-butyl-4-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}(1,4-dioxan-2-ylmethyl)amine
4-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-N-methyl-1,3-thiazol-2-amine
3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]urea
2-(4-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methyl-N-(propan-2-yl)benzamide
1-(cyclopropylmethyl)-5-(quinoxaline-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-[(3-butanamidophenyl)formamido]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
N3-cyclooctyl-N5-(3-methylbutyl)-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1H-1,3-benzodiazole-5-carboxamide
2-ethyl-8-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[5-(3-cyclohexylpyrrolidine-1-carbonyl)-2-methoxyphenoxy]-1-(propan-2-yl)piperidine
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-(5-methyl-1,2-oxazole-4-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
(2S,4R)-N-ethyl-1-(naphthalen-1-ylmethyl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-methyl-6-(piperidin-3-yl)-N-[2-(pyridine-2-sulfonyl)ethyl]pyrimidin-4-amine
[2-ethoxy-5-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)phenyl]methyl acetate
N-{4-[5-(2-aminoethyl)-2-methoxyphenyl]phenyl}acetamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(2,5-difluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
7-(cyclohexylmethyl)-2-(3-methoxypropanoyl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-methyl-1-benzofuran-5-carboxamide
1-(2,3-dihydro-1H-inden-5-yl)-3-methyl-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1H-1,2,4-triazole
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]benzamide
3-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-6-(trifluoromethyl)pyridin-2-ol
1-[4-(4-{[(1-phenylcyclohexyl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
8-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-(2-methoxyethyl)benzamide
3,3-dimethyl-1-{[5-(2-methylpentyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-methyl-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-1,2,3-thiadiazole-5-carboxamide
2-methoxy-1-{1'-[2-(methylsulfanyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
3-(4-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)propanamide
(1S,5R)-3-[(2-chloro-6-fluorophenyl)methyl]-3,9-diazabicyclo[3.3.2]decan-10-one
(5S)-5-{[benzyl({[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
2-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
2-{5-[(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)methyl]-1-[(4-methylphenyl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
7-[(4-fluorophenyl)methyl]-2-(4,4,4-trifluorobutyl)-2,7-diazaspiro[4.5]decan-6-one
1-(2-{1-[2-(4-fluorophenoxy)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}piperidin-1-yl)ethan-1-one
2-[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-4-carboxamide
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-3-propyl-1H-pyrazole-4-carboxamide
{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
2-[ethyl(oxan-4-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[3-(benzyloxy)piperidine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
4-[({2-ethyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)amino]-1-phenylpyrrolidin-2-one
3-hydroxy-3-phenyl-N-[2-(propylsulfanyl)phenyl]pyrrolidine-1-carboxamide