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3-[(2-fluoro-3-methylphenyl)methyl]-4-(hydroxymethyl)-1,3-oxazolidin-2-one
methyl (2S,4R)-4-[3-(4-methylphenyl)propanamido]-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxylate
(1S,5R)-6-(2-ethylpyridine-4-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-(1,2,4-oxadiazol-3-yl)-1-(2-phenylpropyl)piperidine
ethyl 3-[(3-chlorophenyl)methyl]-1-[3-(methylsulfanyl)propanoyl]piperidine-3-carboxylate
1-{6-[4-(pyrazin-2-yl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}azepane
4-(2-methoxyethyl)-1-(3-phenylbutyl)-1,4-diazepan-5-one
N-[(3S,4R)-4-(propan-2-yl)-1-[3-(pyridin-2-yl)propanoyl]pyrrolidin-3-yl]methanesulfonamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(methylsulfanyl)pyridine-3-carboxamide
2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
(4aS,7aR)-1-(2-oxopropanoyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(3aS,6aS)-2-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanoyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-({1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-2-yl}methyl)morpholine
3-[4-(3-phenyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-1,2-benzothiazole
4-(4-{[(1S)-1-(3-methylpyridin-2-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
2-methyl-2-(2-{methyl[(1-methylpyrrolidin-2-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
N,2-dimethyl-2-(morpholin-4-yl)-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
1-[1-(pyrimidin-2-yl)piperidin-4-yl]piperidin-3-ol
(2S)-1-{4-[(2,2-difluoroethyl)carbamoyl]benzenesulfonyl}pyrrolidine-2-carboxylic acid
2-{2-[4-(dimethylamino)piperidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
N-(2-hydroxyethyl)-3-[5-(quinoxalin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
3,3-dimethyl-1-({5-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
4-(4-ethoxy-3-methylphenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-oxobutanamide
4-(carbamoylmethoxy)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
[(3R,4R)-1-[(3-chlorophenyl)methyl]-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
11-{[(5-methylpyrazin-2-yl)methyl]amino}-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-(1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)thiomorpholine
3-(1H-pyrazol-4-yl)-N-[2-(pyridin-3-ylformamido)ethyl]benzamide
4-chloro-N-methyl-3-[({[1-(phenoxymethyl)cyclopropyl]methyl}carbamoyl)amino]benzamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-7-chloro-3,5-dimethyl-1-benzofuran-2-carboxamide
5-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyrazin-2-ol
5-acetyl-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]thiophene-3-carboxamide
(2R)-2-amino-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-methylpentanamide
2-(4-fluorobutyl)-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
3-chloro-2-(3-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-[1-(thiophen-2-yl)ethyl]acetamide
(3S,4R)-1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
4-methyl-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1,3-oxazole-5-carboxamide
3-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}-5,6,7-trimethoxy-1,2-dihydroquinolin-2-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-phenyl-N-(pyridin-3-ylmethyl)propanamide
2-methoxy-1-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
6-tert-butyl-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(1-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-fluorobenzamide
(2S,4S)-N-ethyl-4-[(3E)-hex-3-enamido]-1-(4-methylpyrimidine-5-carbonyl)pyrrolidine-2-carboxamide
N4-{2-[cyclopentyl(methyl)amino]ethyl}-N4,5-dimethylpyrimidine-2,4-diamine
1-(piperidin-1-yl)-3-[2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxy]propan-2-ol
6-fluoro-2-{[4-(1-methoxypropan-2-yl)piperidin-1-yl]methyl}quinolin-4-ol
(4aS,7aR)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione