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3-(5-{[(furan-2-ylmethyl)carbamoyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
1-(5-chloro-3-methyl-1H-indole-2-carbonyl)-4-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,4-diazepan-5-one
5-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-1H-indole
(3S,4R)-1-[2-(2,5-dimethylphenyl)acetyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-[4-(2-methylphenoxy)piperidine-1-carbonyl]cyclopropane-1-carboxamide
5-[4-(4-acetylphenyl)piperazine-1-carbonyl]-1-(cyclohexylmethyl)-N-ethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-(cyclopropylmethyl)-5-(1H-indole-3-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(4-fluorophenyl)-N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
(5-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]propanamide
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
3-[2-(2-methylphenyl)ethyl]piperidine
N-(2-hydroxybutyl)-5-methyl-4-[(2-phenylethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-3-(2-oxooxolan-3-yl)propanamide
3-(4-methyl-1,3-thiazol-5-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)propanamide
N-(2-methoxyethyl)-3-(pyridin-4-yl)-N-(thiophen-3-ylmethyl)propanamide
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
2-(2,5-dimethoxyphenyl)-2-[4-(2-hydroxyphenyl)piperazin-1-yl]acetic acid
N-{[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-(pyridin-3-yl)propanamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxamide
[(1S,3S,3aS,6aR)-3-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
2-[4-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl]acetic acid
N-(isoquinolin-5-ylmethyl)-N,6-dimethyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
3-(2-methoxyethyl)-1-[3-(1H-pyrazol-4-yl)propanoyl]piperidine-3-carboxylic acid
2-[4-(propan-2-yl)morpholin-2-yl]-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
9-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
8-{[(3-fluorophenyl)methyl]carbamoyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-{3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]phenyl}-1,2,3-thiadiazole-4-carboxamide
4-(2-cyclopentylacetyl)-1-(2-methylphenyl)piperazin-2-one
2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-N-(1-methyl-1H-pyrazol-4-yl)acetamide
1-(7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(morpholin-4-yl)propan-1-one
3-{9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}propanoic acid
7-(cyclohexylmethyl)-2-(4-methyl-1,3-thiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-ethyl-3-({2-[3-(furan-2-yl)phenyl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole
N-[(4-fluorophenyl)methyl]-3-[3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-9-yl]propanamide
1-(4-methoxyphenyl)-4-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperazin-2-one
N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(4-chloro-1H-pyrazol-1-yl)propan-1-one
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-[(1-ethylpiperidin-3-yl)methyl]piperidine
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}piperidine
N-[7-methoxy-2-oxo-4-(4-oxo-4H-chromen-3-yl)-1,2,3,4-tetrahydroquinolin-6-yl]acetamide
5-propyl-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-1,2-oxazole-3-carboxamide
2-[4-(3-methylfuran-2-carbonyl)piperazin-1-yl]-1,3-benzoxazole
3-fluoro-N-(1-{1-[6-(propan-2-yl)pyridazin-3-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-(2,3-dimethylphenyl)-9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(3-fluorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
(3R)-3-hydroxy-N-{2-[2-(pyridin-2-yl)ethoxy]phenyl}pyrrolidine-1-carboxamide
methyl 2-(2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamido)acetate
methyl[(4-propyl-4H-1,2,4-triazol-3-yl)methyl][(2,3,4-trifluorophenyl)methyl]amine
1-[4-({2-[(4-methoxyphenyl)methyl]morpholin-4-yl}methyl)thiophen-2-yl]ethan-1-one