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3-(2,4-difluorophenyl)-1-[2-(dimethylamino)ethyl]-6-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-[(4aR,8aS)-6-[4-(trifluoromethyl)benzoyl]-decahydro-1,6-naphthyridine-1-carbonyl]-2-methyl-1,2-dihydrophthalazin-1-one
1-[(4-chlorophenyl)methyl]-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(2-{7-[(2,3-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-(4-fluorophenyl)acetamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
3-[2-(6-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-butyl-2-{2-[(3,3-dimethylpyrrolidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
3-({4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}methyl)pyrrolidin-3-ol
N-{2-[2-(4-fluoro-2-methylphenyl)-1H-imidazol-1-yl]ethyl}-N-methylmethanesulfonamide
4-[3-({1-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperidin-4-yl}oxy)benzoyl]morpholine
5-benzyl-5-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}imidazolidine-2,4-dione
8-(1-hydroxypropan-2-yl)-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 4-[5-({[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
2-methoxy-1-{1'-[1-(propan-2-yl)pyrrolidine-3-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
7-(cyclopropylmethyl)-2-(2,3-dimethylquinoxaline-6-carbonyl)-2,7-diazaspiro[4.5]decane
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
2,5-dimethoxy-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzamide
(4aS,8aS)-2-cyclohexyl-7-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
methyl 2-(1-{[3-(trifluoromethyl)phenyl]carbamoyl}pyrrolidin-3-yl)acetate
14-(6-chloro-2H-1,3-benzodioxol-5-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
1-benzyl-4-[4-(3-methoxyphenyl)-5-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl]piperidine
1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-4-(1,3-thiazol-2-yl)piperazine
(2,1,3-benzoxadiazol-4-ylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
6-(4-ethylphenyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-methoxy-1-{4-[4-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}propan-1-one
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-N'-(2,4-dimethylphenyl)ethanediamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[2-(2,5-dimethylphenoxy)ethyl]-N-methylacetamide
5-[(4-benzylpiperidin-1-yl)methyl]-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
(2E)-N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-3-(thiophen-2-yl)prop-2-enamide
4-[(2-methoxyethyl)amino]-N,5-dimethyl-N-(1,3-thiazol-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
1'-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
methyl[1-(pyrazin-2-yl)propan-2-yl](quinolin-4-ylmethyl)amine
{[4-(methylsulfanyl)phenyl]methyl}(propyl)(pyridin-4-ylmethyl)amine
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-1H-indole-6-carboxamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(oxolan-2-ylmethyl)propanamide
6-(methoxymethyl)-1-methyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
6-[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide
N-{[2-(dimethylamino)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]propanamide
1-(2-methoxyethyl)-N-[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]pyrrolidine-3-carboxamide
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
3-(5-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
N-(2,4-difluorophenyl)-4-{[methyl(pyrazin-2-ylmethyl)amino]methyl}benzamide
2-acetyl-8-(5-propylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{9-[2-(3-methylphenyl)acetyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
2-(3-chloro-4-hydroxyphenyl)-1-{2,7-diazaspiro[4.5]decan-7-yl}ethan-1-one
N-[3-(aminomethyl)phenyl]-4-(4-methoxyphenoxymethyl)piperidine-1-carboxamide
2-methyl-N-[2-(propane-2-sulfonyl)ethyl]-5-sulfamoylbenzamide
2,7,8-trimethyl-4-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]quinoline
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-(5-propylpyrimidin-4-yl)piperidin-4-amine