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6-[3-(2-methylpropoxy)phenyl]pyrazine-2-carboxylic acid
3-[1-(2-methoxyacetyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
4-amino-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyridine-2-carboxamide
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]propanamide
(1S,5R)-3-[2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)acetyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(4S)-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-phenyl-1,3-oxazolidin-2-one
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
(3R,9aR)-3-[(1S)-1-hydroxyethyl]-8-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(azocan-1-yl)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5-[(methylsulfanyl)methyl]furan-2-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(phenylamino)pyrimidine-5-carboxamide
3-[1-(cyclopent-3-ene-1-carbonyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
2-[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-6-methylpyridine-3-carboxylic acid
N-{3-hydroxy-1-[4-(propan-2-yl)phenyl]propyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-[(1-benzylpiperidin-4-yl)methyl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-methylacetamide
[1-(4-methyl-1H-imidazole-5-carbonyl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
2-amino-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-1,3-benzothiazole-5-carboxamide
5-({2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}methyl)-2-(pyrrolidin-1-yl)pyrimidine
5-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-sulfonyl]-2,3-dihydro-1,3-benzoxazol-2-one
2-{[(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl)oxy]methyl}pyridine
3-[1-(isoquinolin-5-ylmethyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-5-ethylpyrimidin-2-amine
N-[1-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopentanecarboxamide
N-[2-(1H-imidazol-1-yl)propyl]-3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propanamide
2-[1-(2-phenylethyl)-4-(quinolin-8-ylmethyl)piperazin-2-yl]ethan-1-ol
1-(3,4-difluorophenyl)-3-[3-(methylsulfanyl)propyl]urea
(2S)-2-amino-1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(1H-imidazol-4-yl)propan-1-one
4-[3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanoyl]piperazine-1-carboxamide
5-(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)-5-propylimidazolidine-2,4-dione
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
1-cyclopentyl-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[2-(pyrazin-2-yl)ethyl]benzamide
4-(1-acetylpiperidin-4-yl)-9-(cyclopropylmethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-{[5-(2-ethoxyethyl)-1-(4-fluorophenyl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
1-ethyl-4-[3-(pyridin-4-yl)azetidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-acetyl-8-[(5-cyano-1-ethyl-1H-pyrrol-3-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N-[(1-methylpyrrolidin-3-yl)methyl]pyrimidin-2-amine
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
1-ethyl-4-{[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-pyrazole
5-(2-fluorophenoxymethyl)-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-pyrazole-3-carboxamide
2-{4-chloro-2-methoxy-6-[(4-methylpiperazin-1-yl)methyl]phenoxy}propanoic acid
(4aS,7aR)-1-[(2-ethylphenyl)methyl]-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(5-methoxy-2-methylphenyl)-7-methyl-2,7-diazaspiro[4.4]nonane-2-carboxamide
1-(furan-2-ylmethyl)-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}piperidine-4-carboxamide
dimethyl(2-{[(5-methylthiophen-2-yl)methyl]({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl})amino}ethyl)amine
3-(4-chloro-1H-pyrazol-1-yl)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}propan-1-one
2-{2-methyl-6-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]pyrimidin-4-yl}ethan-1-amine
2-{[5-(furan-2-yl)-4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid