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N-cyclohexyl-2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
N-[2-(2-chloro-6-fluorophenyl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{5-[2-(1H-imidazol-2-yl)phenyl]-3-methyl-1H-1,2,4-triazol-1-yl}acetic acid
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
(2E)-N-{[3-methyl-7-(1,2,5-thiadiazole-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
5-methyl-6-(4-methylpiperazine-1-carbonyl)-N-[1-(thiophen-2-yl)propyl]thieno[2,3-d]pyrimidin-4-amine
N-[(2R,3R)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-5-fluoro-1-methyl-1H-indole-2-carboxamide
4-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}-1H-indole
N-(3-fluorophenyl)-1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidin-3-amine
2-[1-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
2-{[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-5-methoxy-4H-pyran-4-one
3-{2-[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
methyl (2S,4R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
(4aS,8aR)-6-(2-aminoethyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
7-(cyclopropylmethyl)-2-(1,4-dithiepan-6-yl)-2,7-diazaspiro[4.5]decan-6-one
4-[2-(4-fluorophenyl)piperidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
5-[(4-benzylpiperidin-1-yl)methyl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
2-(1-methyl-1H-pyrrole-2-carbonyl)-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
4-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2-oxazole-3-carboxamide
N3-[3-(2-ethoxyphenyl)propyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
N-(2-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}quinolin-6-yl)acetamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3-(3-hydroxyquinoxalin-2-yl)propanamide
8-(3-fluoropyridin-2-yl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
5-(2,5-dimethylphenoxymethyl)-3-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-oxazole
4-(1-butyl-5-{[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazol-3-yl)benzamide
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
1-{1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]piperidin-3-yl}pyrrolidin-2-one
N-[2-methyl-1-(morpholin-4-yl)propan-2-yl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(methoxymethyl)-1-({2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}sulfonyl)pyrrolidine
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}propanamide
N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}morpholine-2-carboxamide
(3R,4R)-3-methyl-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-4-(oxan-4-yl)piperidin-4-ol
N-[4-(4-{[1-(1,3-thiazol-5-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]pyrazine-2-carboxamide
1-(4-{[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]amino}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-(1-propylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
N-(3-methoxypropyl)-2-(2-methyl-1,3-thiazol-4-yl)-N-[(4-methylphenyl)methyl]acetamide
2-methyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
(3S)-1-ethyl-3-methyl-4-{6-[(thiophen-2-ylmethyl)amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}piperazin-2-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-fluoro-N-methyl-5-sulfamoylbenzamide
N-[4-ethoxy-3-(trifluoromethyl)phenyl]-3-(4H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazin-2-yl}ethan-1-ol
2-(4-fluorophenyl)-N-{2-[7-(quinolin-7-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}acetamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
N-(2-methoxyethyl)-3-{[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-[(5-chloro-1H-indol-2-yl)methyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
4-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
N-butyl-N-methyl-3-({[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide