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N-methyl-N-[2-(methylamino)ethyl]-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
3-(4-fluorophenoxymethyl)-1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidine
1-[(3-{[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
4-[1-(3-phenylpropyl)-5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
3,5-dichloro-4-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}pyridine
1-[1-(4,6-dimethylpyridine-3-carbonyl)piperidin-4-yl]piperidin-4-ol
7-(2,2-dimethylpropyl)-2-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-acetyl-8-(isoquinolin-1-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(3-{[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}phenoxy)acetamide
3-[(2R,3R,6R)-5-(1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N,N-dimethyl-7-(morpholine-2-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
7,8-dimethyl-4-(2-methylpiperidine-1-carbonyl)-2-(pyrimidin-5-yl)quinoline
(1S,5R)-6-(1-benzothiophene-2-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2-methoxyethyl)-1-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2-({imidazo[2,1-b][1,3]thiazol-6-ylformamido}methyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-[(6-fluoro-1-methyl-1H-indol-3-yl)methyl]-decahydro-1,6-naphthyridin-2-one
4-[(3S)-3-hydroxy-3-phenylpropyl]-1-(2-methoxyphenyl)piperazin-2-one
1-(3-chlorophenyl)-4-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]piperazine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,3,5-trimethyl-1H-pyrrole-2-carboxamide
1-(2-methoxyphenyl)-2,2-dimethyl-4-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperazine
5-{[(5-chlorothiophen-2-yl)methyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1S,5R)-6-(2-methyl-1,3-thiazole-4-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-cyclopentyl-N-(2-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
5-{2-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-5-methyl-N,N-bis(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
(3R,4S)-4-cyclopropyl-1-[3-(dimethylamino)benzoyl]pyrrolidin-3-amine
2-{4-[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]piperidin-1-yl}pyridine-4-carbonitrile
3-(3-phenylpropyl)-1-(pyrazin-2-yl)piperidine-3-carboxylic acid
5-[2-(cyclobutylamino)pyrimidin-4-yl]-2-ethoxybenzoic acid
5-(6-methoxypyrimidin-4-yl)-1H-indole
N-(3-{2-methoxy-5-[(3-oxopiperazin-1-yl)methyl]phenoxy}propyl)oxolane-2-carboxamide
(2S,3R)-2-amino-1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-hydroxybutan-1-one
N-[3-(3-{[cyclohexyl(methyl)amino]methyl}phenoxy)propyl]-3-methylthiophene-2-carboxamide
4-methoxy-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-3-(morpholin-4-yl)benzamide
ethyl 4-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-amido}piperidine-1-carboxylate
1-[9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
1-ethyl-3-(2-methylpropyl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide
1-{3-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propyl}-5-methyl-1H-1,2,3,4-tetrazole
1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-indole-5-carboxamide
N-[(2-methoxyphenyl)methyl]-1-methyl-N-[(3-methylphenyl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
4-[(dimethylamino)methyl]-N-[1-(pyridin-4-yl)propyl]benzamide
3-(3-methoxyphenoxy)-1-(3-methylthiophene-2-carbonyl)azetidine
4-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
N-{1-[(2-ethylpyrimidin-5-yl)methyl]azepan-4-yl}benzenesulfonamide
4-(3,5-difluoro-2-methoxyphenyl)thiophene-2-carboxamide
N,3-dimethyl-5-(phenoxymethyl)-N-(prop-2-en-1-yl)furan-2-carboxamide
(2R)-2-{[5-(3-acetylphenoxymethyl)-1H-pyrazol-3-yl]formamido}propanamide
4-[(4-methyl-1,3-thiazol-2-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 6-(cyclopent-1-ene-1-carbonyl)-2-[(3-fluorophenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate